# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666534 | Not Active | Homo sapiens | |||||
2. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666533 | Not Active | Homo sapiens | |||||
3. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666532 | Not Active | Homo sapiens | |||||
4. | PROTAC CRBN Degrader-1 | 14a | %max | = | 75 | % | ALA4666531 | % | Homo sapiens | |||
5. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 64 | % | ALA4666531 | % | Homo sapiens | |||
6. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 19 | % | ALA4666530 | % | Homo sapiens | |||
7. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666529 | Not Active | Homo sapiens | |||||
8. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666528 | Active | Homo sapiens | |||||
9. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666527 | Active | Homo sapiens | |||||
10. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 19 | % | ALA4666526 | % | Homo sapiens | |||
11. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 103 | % | ALA4666525 | % | Homo sapiens | |||
12. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 100 | % | ALA4666524 | % | Homo sapiens | |||
13. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 81 | % | ALA4666523 | % | Homo sapiens | |||
14. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 64 | % | ALA4666522 | % | Homo sapiens | |||
15. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 95 | % | ALA4666521 | % | Homo sapiens | |||
16. | PROTAC CRBN Degrader-1 | 14a | DC50 | = | 200 | nM | ALA4666520 | nM | Homo sapiens | |||
17. | PROTAC CRBN Degrader-1 | 14a | Activity | 0 | ALA4666519 | Active | Homo sapiens | |||||
18. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 86 | % | ALA4666518 | % | Homo sapiens | |||
19. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 49 | % | ALA4666517 | % | Homo sapiens | |||
20. | PROTAC CRBN Degrader-1 | 14a | Activity | = | 25 | % | ALA4666516 | % | Homo sapiens |