| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4763134 | 15 | Emax | = | 9 | % | ALA4701636 | % | Homo sapiens | |||
| 2. | ALA4763134 | 15 | INH | = | 77 | % | ALA4701634 | % | Mus musculus | |||
| 3. | ALA4763134 | 15 | INH | = | 50 | % | ALA4701633 | % | Mus musculus | |||
| 4. | ALA4763134 | 15 | INH | = | 39 | % | ALA4701632 | % | Mus musculus | |||
| 5. | ALA4763134 | 15 | F | = | 100 | % | ALA4701629 | % | ||||
| 6. | ALA4763134 | 15 | t1/2 | = | 27 | hr | ALA4701628 | hr | ||||
| 7. | ALA4763134 | 15 | Vdss | = | 1.2 | L/Kg | ALA4701627 | L.kg-1 | ||||
| 8. | ALA4763134 | 15 | CL | = | 1.1 | ml/min.kg | ALA4701626 | mL.min-1.kg-1 | ||||
| 9. | ALA4763134 | 15 | AUC | = | 55 | uM.hr | ALA4701625 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 10. | ALA4763134 | 15 | AUC | = | 23 | uM.hr | ALA4701624 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 11. | ALA4763134 | 15 | Cmax | = | 3.9 | uM | ALA4701623 | nM | ||||
| 12. | ALA4763134 | 15 | F | = | 90 | % | ALA4701622 | % | ||||
| 13. | ALA4763134 | 15 | t1/2 | = | 28 | hr | ALA4701621 | hr | ||||
| 14. | ALA4763134 | 15 | Vdss | = | 0.7 | L/Kg | ALA4701620 | L.kg-1 | ||||
| 15. | ALA4763134 | 15 | CL | = | 0.3 | ml/min.kg | ALA4701619 | mL.min-1.kg-1 | ||||
| 16. | ALA4763134 | 15 | AUC | = | 144 | uM.hr | ALA4701618 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 17. | ALA4763134 | 15 | AUC | = | 80 | uM.hr | ALA4701617 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 18. | ALA4763134 | 15 | Cmax | = | 3.8 | uM | ALA4701616 | nM | ||||
| 19. | ALA4763134 | 15 | F | = | 100 | % | ALA4701615 | % | ||||
| 20. | ALA4763134 | 15 | t1/2 | = | 5.8 | hr | ALA4701614 | hr |
The page will load shortly, Thanks for your patience!