# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4763327 | 27 | IC50 | = | 0.536 | uM | ALA4673830 | 6.27 | nM | Homo sapiens | ||
2. | ALA4763327 | 27 | EC50 | > | 100 | uM | ALA4673829 | nM | Homo sapiens | |||
3. | ALA4763327 | 27 | logD | = | 2.6 | ALA4673828 | ||||||
4. | ALA4763327 | 27 | CLH | = | 35 | microL/min/mg | ALA4673827 | mL.min-1.g-1 | ||||
5. | ALA4763327 | 27 | Fu | = | 11 | % | ALA4673826 | |||||
6. | ALA4763327 | 27 | permeability | = | 5.2 | 10^-6 cm/s | ALA4673825 | 10^-6 cm/s | ||||
7. | ALA4763327 | 27 | F | = | 31 | % | ALA4673823 | % | ||||
8. | ALA4763327 | 27 | CL | = | 29 | ml/min.kg | ALA4673822 | mL.min-1.kg-1 | ||||
9. | ALA4763327 | 27 | Vdss | = | 1.1 | L/Kg | ALA4673821 | L.kg-1 | ||||
10. | ALA4763327 | 27 | t1/2 | = | 1.2 | hr | ALA4673819 | hr | ||||
11. | ALA4763327 | 27 | Kd | = | 0.44 | uM | ALA4673817 | 6.36 | nM | Homo sapiens | ||
12. | ALA4763327 | 27 | EC50 | = | 1.5 | uM | ALA4673815 | 5.82 | nM | Homo sapiens |