# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4776259 | 21i; S15 | IC50 | = | 29 | nM | ALA4676505 | 7.54 | nM | Homo sapiens | ||
2. | ALA4776259 | 21i; S15 | IC50 | = | 375 | nM | ALA4676504 | 6.43 | nM | Homo sapiens | ||
3. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676503 | nM | Homo sapiens | |||
4. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676502 | nM | ||||
5. | ALA4776259 | 21i; S15 | Activity | = | 14 | % | ALA4676501 | % | Homo sapiens | |||
6. | ALA4776259 | 21i; S15 | Activity | = | 176 | % | ALA4676500 | % | Homo sapiens | |||
7. | ALA4776259 | 21i; S15 | INH | = | 77 | % | ALA4676498 | % | Homo sapiens | |||
8. | ALA4776259 | 21i; S15 | INH | = | 13 | % | ALA4676497 | % | Homo sapiens | |||
9. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676496 | nM | Rattus norvegicus | |||
10. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676495 | nM | Homo sapiens | |||
11. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676494 | nM | Homo sapiens | |||
12. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676493 | nM | Homo sapiens | |||
13. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676491 | nM | Homo sapiens | |||
14. | ALA4776259 | 21i; S15 | INH | = | 98 | % | ALA4676490 | % | Homo sapiens | |||
15. | ALA4776259 | 21i; S15 | INH | = | 67 | % | ALA4676489 | % | Homo sapiens | |||
16. | ALA4776259 | 21i; S15 | Activity | = | 8 | % | ALA4676487 | % | Homo sapiens | |||
17. | ALA4776259 | 21i; S15 | IC50 | > | 5000 | nM | ALA4676486 | nM | Homo sapiens | |||
18. | ALA4776259 | 21i; S15 | Ratio IC50 | = | 13 | ALA4676480 | ||||||
19. | ALA4776259 | 21i; S15 | 2aPTT | = | 236 | uM | ALA4676479 | uM | Homo sapiens | |||
20. | ALA4776259 | 21i; S15 | TDI | 0 | ALA4676478 | Active | Homo sapiens |