# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4776685 | Cpd E | IC50 | = | 1.9 | nM | ALA4669389 | 8.72 | nM | Homo sapiens | ||
2. | ALA4776685 | Cpd E | IC50 | = | 2.5 | nM | ALA4669388 | 8.60 | nM | Homo sapiens | ||
3. | ALA4776685 | Cpd E | IC50 | = | 18.1 | nM | ALA4669387 | 7.74 | nM | Homo sapiens | ||
4. | ALA4776685 | Cpd E | IC50 | = | 9829 | nM | ALA4669386 | 5.01 | nM | Homo sapiens | ||
5. | ALA4776685 | Cpd E | IC50 | = | 5422 | nM | ALA4669385 | 5.27 | nM | Homo sapiens | ||
6. | ALA4776685 | Cpd E | EC50 | = | 294 | nM | ALA4669384 | 6.53 | nM | Homo sapiens | ||
7. | ALA4776685 | Cpd E | EC50 | = | 269 | nM | ALA4669383 | 6.57 | nM | Homo sapiens | ||
8. | ALA4776685 | Cpd E | CL free | = | 166 | ml/min.kg | ALA4669382 | mL.min-1.kg-1 | ||||
9. | ALA4776685 | Cpd E | Vdu | = | 45 | L/Kg | ALA4669381 | L.kg-1 | ||||
10. | ALA4776685 | Cpd E | t1/2 | = | 6.4 | hr | ALA4669380 | hr | ||||
11. | ALA4776685 | Cpd E | F | = | 0 | % | ALA4669379 | % | ||||
12. | ALA4776685 | Cpd E | Papp | = | 1.1 | 10^-6 cm/s | ALA4669377 | 10^-6 cm/s | ||||
13. | ALA4776685 | Cpd E | EC50 | = | 269 | nM | ALA4813309 | 6.57 | nM | Human immunodeficiency virus | ||
14. | ALA4776685 | Cpd E | EC50 | = | 294 | nM | ALA4813308 | 6.53 | nM | Human immunodeficiency virus | ||
15. | ALA4776685 | Cpd E | IC50 | = | 5422 | nM | ALA4813307 | 5.27 | nM | Homo sapiens | ||
16. | ALA4776685 | Cpd E | IC50 | = | 9829 | nM | ALA4813306 | 5.01 | nM | Homo sapiens | ||
17. | ALA4776685 | Cpd E | IC50 | = | 2.5 | nM | ALA4813305 | 8.60 | nM | Homo sapiens | ||
18. | ALA4776685 | Cpd E | IC50 | = | 18 | nM | ALA4813304 | 7.75 | nM | Homo sapiens | ||
19. | ALA4776685 | Cpd E | IC50 | = | 1.9 | nM | ALA4813303 | 8.72 | nM | Homo sapiens |