| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4776839 | 3; BI-0252 | Vdss | = | 2.1 | L/Kg | ALA4681457 | L.kg-1 | ||||
| 2. | ALA4776839 | 3; BI-0252 | CL | = | 7.1 | ml/min.kg | ALA4681456 | mL.min-1.kg-1 | ||||
| 3. | ALA4776839 | 3; BI-0252 | Cmax | = | 21.3 | uM | ALA4681455 | nM | ||||
| 4. | ALA4776839 | 3; BI-0252 | AUC | = | 264 | uM.hr | ALA4681454 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 5. | ALA4776839 | 3; BI-0252 | IC50 | > | 25000 | nM | ALA4681453 | nM | Homo sapiens | |||
| 6. | ALA4776839 | 3; BI-0252 | IC50 | = | 471 | nM | ALA4681452 | 6.33 | nM | Homo sapiens | ||
| 7. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681451 | Active | % | |||||
| 8. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681450 | Active | % | |||||
| 9. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681449 | Active | % | |||||
| 10. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681448 | Active | % | |||||
| 11. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681447 | Active | % | |||||
| 12. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681446 | Active | % | |||||
| 13. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681445 | Tde | % | |||||
| 14. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681444 | Tde | % | |||||
| 15. | ALA4776839 | 3; BI-0252 | INH | 0 | ALA4681443 | Tde | % | |||||
| 16. | ALA4776839 | 3; BI-0252 | Activity | 0 | ALA4681442 | Active | Homo sapiens | |||||
| 17. | ALA4776839 | 3; BI-0252 | Activity | 0 | ALA4681441 | Active | Homo sapiens | |||||
| 18. | ALA4776839 | 3; BI-0252 | IC50 | = | 4 | nM | ALA4681440 | 8.40 | nM | Homo sapiens |
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