| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4777187 | 8 | IC50 | = | 90 | uM | ALA4673991 | 4.05 | nM | Mus musculus | ||
| 2. | ALA4777187 | 8 | LD50 | > | 2000 | mg kg-1 | ALA4673990 | mg.kg-1 | ||||
| 3. | ALA4777187 | 8 | Activity | = | 11.58 | mmol/L | ALA4673979 | mmol/L | Mus musculus | |||
| 4. | ALA4777187 | 8 | Activity | = | 29.83 | umol/L | ALA4673978 | umol/L | Mus musculus | |||
| 5. | ALA4777187 | 8 | Activity | = | 222.92 | uL/min | ALA4673977 | uL/min | Mus musculus | |||
| 6. | ALA4777187 | 8 | Activity | = | 41.96 | ug | ALA4673976 | ug | Mus musculus | |||
| 7. | ALA4777187 | 8 | Activity | = | 0.37 | ug/mg | ALA4673975 | ug/mg | Mus musculus | |||
| 8. | ALA4777187 | 8 | Activity | = | 67.31 | % | ALA4673972 | % | Mus musculus | |||
| 9. | ALA4777187 | 8 | Activity | 0 | ALA4673971 | Active | Rattus norvegicus | |||||
| 10. | ALA4777187 | 8 | Activity | 0 | ALA4673969 | Active | Rattus norvegicus | |||||
| 11. | ALA4777187 | 8 | Activity | 0 | ALA4673968 | Active | Rattus norvegicus | |||||
| 12. | ALA4777187 | 8 | Activity | 0 | ALA4673967 | Active | ||||||
| 13. | ALA4777187 | 8 | Activity | 0 | ALA4673966 | Active | ||||||
| 14. | ALA4777187 | 8 | FC | = | 1.85 | ALA4673965 | ||||||
| 15. | ALA4777187 | 8 | FC | = | 2.42 | ALA4673964 | ||||||
| 16. | ALA4777187 | 8 | t1/2 | = | 4.89 | hr | ALA4673958 | hr | ||||
| 17. | ALA4777187 | 8 | Cmax | = | 2032 | ng/ml | ALA4673957 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 18. | ALA4777187 | 8 | AUCt | = | 11214.77 | hr.ng/ml | ALA4673956 | ng.hr.mL-1 | ||||
| 19. | ALA4777187 | 8 | solubility | 0 | ALA4673952 | Soluble | ||||||
| 20. | ALA4777187 | 8 | permeability | 0 | ALA4673951 | Permeable |
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