# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4777230 | 23 | Activity | 0 | ALA4689190 | Not Active | Mus musculus | |||||
2. | ALA4777230 | 23 | Activity | 0 | ALA4689189 | Not Active | Mus musculus | |||||
3. | ALA4777230 | 23 | AUC | = | 38 | uM.hr | ALA4689188 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
4. | ALA4777230 | 23 | Drug uptake | = | 0.06 | uM | ALA4689187 | uM | ||||
5. | ALA4777230 | 23 | Drug uptake | = | 1.9 | uM | ALA4689186 | uM | ||||
6. | ALA4777230 | 23 | Cmax | = | 9.3 | uM | ALA4689185 | nM | ||||
7. | ALA4777230 | 23 | Ratio | = | 0.3 | ALA4689184 | ||||||
8. | ALA4777230 | 23 | permeability | = | 73 | nm/s | ALA4689183 | nm/s | ||||
9. | ALA4777230 | 23 | Stabilty | = | 85 | % | ALA4689182 | % | ||||
10. | ALA4777230 | 23 | Stabilty | = | 85 | % | ALA4689181 | % | ||||
11. | ALA4777230 | 23 | Stabilty | = | 76 | % | ALA4689180 | % | ||||
12. | ALA4777230 | 23 | EC50 | = | 34 | nM | ALA4689176 | 7.47 | nM | Mus musculus | ||
13. | ALA4777230 | 23 | EC50 | = | 25 | nM | ALA4689175 | 7.60 | nM | Homo sapiens | ||
14. | ALA4777230 | 23 | EC50 | = | 15 | nM | ALA4689173 | 7.82 | nM | Homo sapiens |