| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4778264 | 11 | pKa | = | 1.9 | ALA4766401 | ||||||
| 2. | ALA4778264 | 11 | Activity | 0 | ALA4766302 | Not Active | Homo sapiens | |||||
| 3. | ALA4778264 | 11 | Activity | 0 | ALA4766301 | Not Active | Homo sapiens | |||||
| 4. | ALA4778264 | 11 | Activity | 0 | ALA4766300 | Not Active | Homo sapiens | |||||
| 5. | ALA4778264 | 11 | PPB | > | 99 | % | ALA4766299 | % | ||||
| 6. | ALA4778264 | 11 | ED90 | > | 100 | mg kg-1 | ALA4766284 | mg kg-1 | Mus musculus | |||
| 7. | ALA4778264 | 11 | Activity | 0 | ALA4766283 | Not Active | Mus musculus | |||||
| 8. | ALA4778264 | 11 | Time | = | 4.7 | min | ALA4766282 | hr | Homo sapiens | |||
| 9. | ALA4778264 | 11 | Kd | = | 37 | nM | ALA4766281 | 7.43 | nM | Homo sapiens | ||
| 10. | ALA4778264 | 11 | Emax | = | 124 | % | ALA4766280 | % | Homo sapiens | |||
| 11. | ALA4778264 | 11 | EC50 | = | 68 | nM | ALA4766279 | 7.17 | nM | Homo sapiens | ||
| 12. | ALA4778264 | 11 | Emax | = | 61 | % | ALA4766278 | % | Rattus norvegicus | |||
| 13. | ALA4778264 | 11 | EC50 | = | 14000 | nM | ALA4766277 | 4.85 | nM | Rattus norvegicus | ||
| 14. | ALA4778264 | 11 | Emax | = | 98 | % | ALA4766276 | % | Mus musculus | |||
| 15. | ALA4778264 | 11 | EC50 | = | 3800 | nM | ALA4766275 | 5.42 | nM | Mus musculus | ||
| 16. | ALA4778264 | 11 | Emax | = | 141 | % | ALA4766274 | % | Homo sapiens | |||
| 17. | ALA4778264 | 11 | EC50 | = | 600 | nM | ALA4766273 | 6.22 | nM | Homo sapiens | ||
| 18. | ALA4778264 | 11 | Emax | = | 54 | % | ALA4766272 | % | Homo sapiens | |||
| 19. | ALA4778264 | 11 | EC50 | = | 14 | nM | ALA4766271 | 7.85 | nM | Homo sapiens | ||
| 20. | ALA4778264 | 11 | Ki | = | 79 | nM | ALA4766270 | 7.10 | nM | Homo sapiens |
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