# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4778548 | 8; BI-0319 | pIC50 | = | 7.7 | ALA4675423 | 7.70 | nM | Homo sapiens | |||
2. | ALA4778548 | 8; BI-0319 | IC50 | = | 19 | nM | ALA4675423 | 7.72 | nM | Homo sapiens | ||
3. | ALA4778548 | 8; BI-0319 | pDC50 | = | 6.7 | ALA4675421 | Homo sapiens | |||||
4. | ALA4778548 | 8; BI-0319 | Emax | = | 80 | % | ALA4675419 | % | Homo sapiens | |||
5. | ALA4778548 | 8; BI-0319 | Activity | 0 | ALA4675416 | Not Active | Homo sapiens | |||||
6. | ALA4778548 | 8; BI-0319 | INH | > | 90 | % | ALA4675414 | % | Homo sapiens | |||
7. | ALA4778548 | 8; BI-0319 | INH | > | 90 | % | ALA4675413 | % | Homo sapiens | |||
8. | ALA4778548 | 8; BI-0319 | INH | > | 90 | % | ALA4675412 | % | Homo sapiens | |||
9. | ALA4778548 | 8; BI-0319 | Activity | 0 | ALA4675411 | Not Active | ||||||
10. | ALA4778548 | 8; BI-0319 | Activity | 0 | ALA4675410 | Active | Homo sapiens | |||||
11. | ALA4778548 | 8; BI-0319 | Activity | 0 | ALA4675409 | Active | Homo sapiens | |||||
12. | ALA4778548 | 8; BI-0319 | pDC50 | = | 6.2 | ALA4675407 | Homo sapiens | |||||
13. | ALA4778548 | 8; BI-0319 | Emax | = | 59 | % | ALA4675405 | % | Homo sapiens | |||
14. | ALA4778548 | 8; BI-0319 | pDC50 | = | 7.4 | ALA4675403 | Homo sapiens | |||||
15. | ALA4778548 | 8; BI-0319 | Emax | = | 88 | % | ALA4675401 | % | Homo sapiens | |||
16. | ALA4778548 | 8; BI-0319 | Fu | = | 4 | % | ALA4675400 | |||||
17. | ALA4778548 | 8; BI-0319 | permeability | 0 | ALA4675399 | Impermeable | ||||||
18. | ALA4778548 | 8; BI-0319 | Time | = | 20 | hr | ALA4675396 | hr | Homo sapiens | |||
19. | ALA4778548 | 8; BI-0319 | Stabilty | 0 | ALA4675395 | Stable | % | |||||
20. | ALA4778548 | 8; BI-0319 | Time | = | 72 | hr | ALA4675392 | hr | Homo sapiens |