# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | AZ14117230 | 106; PROTAC 1 | pIC50 | = | 8.1 | ALA5137714 | 8.10 | nM | ||||
2. | AZ14117230 | 106; PROTAC 1 | pKd | = | 9 | ALA5137713 | 9.00 | nM | Homo sapiens | |||
3. | AZ14117230 | 106; PROTAC 1 | pIC50 | = | 8.11 | ALA5127898 | 8.11 | nM | Homo sapiens | |||
4. | AZ14117230 | 106; PROTAC 1 | pKd | = | 9.27 | ALA5127897 | 9.27 | nM | Homo sapiens | |||
5. | AZ14117230 | 106; PROTAC 1 | GI50 | = | 57 | nM | ALA5127831 | nM | Homo sapiens | |||
6. | AZ14117230 | 106; PROTAC 1 | Drug uptake | = | 0.79 | pmol | ALA4735370 | pmol | ||||
7. | AZ14117230 | 106; PROTAC 1 | Drug uptake | = | 0.03 | pmol | ALA4735369 | pmol | ||||
8. | AZ14117230 | 106; PROTAC 1 | GI50 | = | 57 | nM | ALA4735368 | nM | Homo sapiens | |||
9. | AZ14117230 | 106; PROTAC 1 | Kd | < | 1 | nM | ALA4735367 | nM | Homo sapiens |