# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4779479 | 22 | INH | > | 65 | % | ALA4714744 | % | Homo sapiens | |||
2. | ALA4779479 | 22 | INH | > | 65 | % | ALA4714743 | % | Homo sapiens | |||
3. | ALA4779479 | 22 | INH | > | 65 | % | ALA4714742 | % | Homo sapiens | |||
4. | ALA4779479 | 22 | INH | > | 65 | % | ALA4714741 | % | Homo sapiens | |||
5. | ALA4779479 | 22 | Ratio | = | 20 | ALA4714740 | ||||||
6. | ALA4779479 | 22 | Papp | = | 20 | 10^-6 cm/s | ALA4714739 | 10^-6 cm/s | ||||
7. | ALA4779479 | 22 | Papp | = | 1 | 10^-6 cm/s | ALA4714738 | 10^-6 cm/s | ||||
8. | ALA4779479 | 22 | t1/2 | > | 2 | hr | ALA4714737 | hr | ||||
9. | ALA4779479 | 22 | t1/2 | > | 2 | hr | ALA4714736 | hr | ||||
10. | ALA4779479 | 22 | t1/2 | > | 2 | hr | ALA4714735 | hr | ||||
11. | ALA4779479 | 22 | solubility | = | 30 | uM | ALA4714734 | nM | ||||
12. | ALA4779479 | 22 | Kd | = | 55 | nM | ALA4714733 | 7.26 | nM | Homo sapiens |