# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4779612 | 19 | Activity | 0 | ALA4767518 | Non-Toxic | ||||||
2. | ALA4779612 | 19 | Activity | 0 | ALA4767517 | Non-Toxic | ||||||
3. | ALA4779612 | 19 | INH | = | 63 | % | ALA4767516 | % | Mus musculus | |||
4. | ALA4779612 | 19 | INH | = | 51 | % | ALA4767515 | % | Mus musculus | |||
5. | ALA4779612 | 19 | INH | = | 65 | % | ALA4767514 | % | Homo sapiens | |||
6. | ALA4779612 | 19 | INH | = | 54 | % | ALA4767513 | % | Homo sapiens | |||
7. | ALA4779612 | 19 | AUC | = | 1124.8 | ng.hr/ml | ALA4767506 | ng.hr.mL-1 | ||||
8. | ALA4779612 | 19 | AUC | = | 1173.5 | ng.hr/ml | ALA4767505 | ng.hr.mL-1 | ||||
9. | ALA4779612 | 19 | t1/2 | = | 7.1 | hr | ALA4767504 | hr | ||||
10. | ALA4779612 | 19 | Vd | = | 21.6 | L/Kg | ALA4767503 | L.kg-1 | ||||
11. | ALA4779612 | 19 | F | = | 7.55 | % | ALA4767502 | % | ||||
12. | ALA4779612 | 19 | Cmax | = | 31.5 | ng/ml | ALA4767490 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
13. | ALA4779612 | 19 | Tmax | = | 0.083 | hr | ALA4767489 | hr | ||||
14. | ALA4779612 | 19 | t1/2 | = | 20.1 | hr | ALA4767488 | hr | ||||
15. | ALA4779612 | 19 | AUC | = | 470.8 | ng.hr/ml | ALA4767487 | ng.hr.mL-1 | ||||
16. | ALA4779612 | 19 | AUC | = | 129.7 | ng.hr/ml | ALA4767486 | ng.hr.mL-1 | ||||
17. | ALA4779612 | 19 | C0 | = | 4130.8 | ng/L | ALA4767475 | ng/L | ||||
18. | ALA4779612 | 19 | CL | = | 2.12 | ml/hr.kg | ALA4767474 | mL.min-1.kg-1 | ||||
19. | ALA4779612 | 19 | Drug metabolism | = | 64.2 | % | ALA4767473 | % | ||||
20. | ALA4779612 | 19 | Stabilty | = | 14 | % | ALA4767472 | % |