| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4780641 | 25 | pKa | = | 8.3 | ALA4766402 | ||||||
| 2. | ALA4780641 | 25 | pKa | = | 4.3 | ALA4766401 | ||||||
| 3. | ALA4780641 | 25 | AUC | = | 1029 | ng.hr/ml | ALA4766397 | ng.hr.mL-1 | ||||
| 4. | ALA4780641 | 25 | Activity | 0 | ALA4766302 | Not Active | Homo sapiens | |||||
| 5. | ALA4780641 | 25 | Activity | 0 | ALA4766301 | Not Active | Homo sapiens | |||||
| 6. | ALA4780641 | 25 | Activity | 0 | ALA4766300 | Not Active | Homo sapiens | |||||
| 7. | ALA4780641 | 25 | PPB | > | 99 | % | ALA4766299 | % | ||||
| 8. | ALA4780641 | 25 | ED90 | = | 11.7 | mg kg-1 | ALA4766284 | mg kg-1 | Mus musculus | |||
| 9. | ALA4780641 | 25 | Activity | 0 | ALA4766283 | Active | Mus musculus | |||||
| 10. | ALA4780641 | 25 | Time | = | 47 | min | ALA4766282 | hr | Homo sapiens | |||
| 11. | ALA4780641 | 25 | Kd | = | 9.5 | nM | ALA4766281 | 8.02 | nM | Homo sapiens | ||
| 12. | ALA4780641 | 25 | Emax | = | 268 | % | ALA4766280 | % | Homo sapiens | |||
| 13. | ALA4780641 | 25 | EC50 | = | 12 | nM | ALA4766279 | 7.92 | nM | Homo sapiens | ||
| 14. | ALA4780641 | 25 | Emax | = | 126 | % | ALA4766278 | % | Rattus norvegicus | |||
| 15. | ALA4780641 | 25 | EC50 | = | 5.5 | nM | ALA4766277 | 8.26 | nM | Rattus norvegicus | ||
| 16. | ALA4780641 | 25 | Emax | = | 131 | % | ALA4766276 | % | Mus musculus | |||
| 17. | ALA4780641 | 25 | EC50 | = | 3.3 | nM | ALA4766275 | 8.48 | nM | Mus musculus | ||
| 18. | ALA4780641 | 25 | Emax | = | 134 | % | ALA4766274 | % | Homo sapiens | |||
| 19. | ALA4780641 | 25 | EC50 | = | 56 | nM | ALA4766273 | 7.25 | nM | Homo sapiens | ||
| 20. | ALA4780641 | 25 | Emax | = | 47 | % | ALA4766272 | % | Homo sapiens |
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