# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4781761 | IIIb; C-2048 | deltaTm | = | 3.9 | degrees C | ALA4773247 | degrees C | ||||
2. | ALA4781761 | IIIb; C-2048 | deltaTm | = | 26.6 | degrees C | ALA4773246 | degrees C | Homo sapiens | |||
3. | ALA4781761 | IIIb; C-2048 | deltaTm | = | 26.1 | degrees C | ALA4773245 | degrees C | Homo sapiens | |||
4. | ALA4781761 | IIIb; C-2048 | deltaTm | = | 33.2 | degrees C | ALA4773244 | degrees C | Homo sapiens | |||
5. | ALA4781761 | IIIb; C-2048 | TGI | = | 39 | % | ALA4773235 | % | Homo sapiens | |||
6. | ALA4781761 | IIIb; C-2048 | T/C | = | 300 | % | ALA4773148 | % | Rattus norvegicus | |||
7. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.033 | uM | ALA4773140 | 7.48 | nM | Homo sapiens | ||
8. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.103 | uM | ALA4773139 | 6.99 | nM | Homo sapiens | ||
9. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.12 | uM | ALA4773138 | 6.92 | nM | Homo sapiens | ||
10. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.041 | uM | ALA4773137 | 7.39 | nM | Homo sapiens | ||
11. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.138 | uM | ALA4773136 | 6.86 | nM | Homo sapiens | ||
12. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.152 | uM | ALA4773135 | 6.82 | nM | Homo sapiens | ||
13. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.022 | uM | ALA4773132 | 7.66 | nM | Homo sapiens | ||
14. | ALA4781761 | IIIb; C-2048 | IC50 | = | 0.022 | uM | ALA4773127 | 7.66 | nM | Homo sapiens |