# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4781940 | 20 | F | = | 21 | % | ALA4669532 | % | ||||
2. | ALA4781940 | 20 | AUC | = | 0.57 | ug.hr/ml | ALA4669531 | ng.hr.mL-1 | ||||
3. | ALA4781940 | 20 | t1/2 | = | 5.5 | hr | ALA4669530 | hr | ||||
4. | ALA4781940 | 20 | Cmax | = | 0.2 | ug/hr | ALA4669529 | ug/hr | ||||
5. | ALA4781940 | 20 | Tmax | = | 2 | hr | ALA4669528 | hr | ||||
6. | ALA4781940 | 20 | Vdss | = | 6.3 | L/Kg | ALA4669527 | L.kg-1 | ||||
7. | ALA4781940 | 20 | CL | = | 1.73 | L/hr/kg | ALA4669526 | mL.min-1.kg-1 | ||||
8. | ALA4781940 | 20 | AUC | = | 1.11 | ug.hr/ml | ALA4669525 | ng.hr.mL-1 | ||||
9. | ALA4781940 | 20 | t1/2 | = | 5.9 | hr | ALA4669524 | hr | ||||
10. | ALA4781940 | 20 | CC50 | > | 100 | uM | ALA4669523 | nM | Cricetulus griseus | |||
11. | ALA4781940 | 20 | CC50 | > | 100 | uM | ALA4669522 | nM | Mus musculus | |||
12. | ALA4781940 | 20 | CC50 | > | 100 | uM | ALA4669521 | nM | Mus musculus | |||
13. | ALA4781940 | 20 | CC50 | > | 100 | uM | ALA4669520 | nM | Homo sapiens | |||
14. | ALA4781940 | 20 | CC50 | > | 100 | uM | ALA4669519 | nM | Chlorocebus sabaeus | |||
15. | ALA4781940 | 20 | Stabilty | = | 56.4 | % | ALA4669518 | % | ||||
16. | ALA4781940 | 20 | Stabilty | = | 60.7 | % | ALA4669517 | % | ||||
17. | ALA4781940 | 20 | Ratio CC50/IC50 | = | 25 | ALA4669516 | ||||||
18. | ALA4781940 | 20 | CC50 | = | 3.59 | uM | ALA4669515 | nM | Chlorocebus sabaeus | |||
19. | ALA4781940 | 20 | IC50 | = | 0.157 | uM | ALA4669514 | 6.80 | nM | Middle East respiratory syndrome-related coronavirus | ||
20. | ALA4781940 | 20 | Activity | > | 50 | uM | ALA4669513 | uM | Homo sapiens |