| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  GPR40 Activator 1 | 18 | pKa | = | 7.4 | ALA4766402 | ||||||
| 2. | GPR40 Activator 1 | 18 | pKa | = | 4.2 | ALA4766401 | ||||||
| 3. | GPR40 Activator 1 | 18 | Drug uptake | 0 | ALA4766308 | Active | ||||||
| 4. | GPR40 Activator 1 | 18 | Drug uptake | 0 | ALA4766307 | Active | ||||||
| 5. | GPR40 Activator 1 | 18 | Drug uptake | 0 | ALA4766306 | Active | ||||||
| 6. | GPR40 Activator 1 | 18 | Drug uptake | 0 | ALA4766305 | Active | ||||||
| 7. | GPR40 Activator 1 | 18 | AUC | = | 1055 | ng.hr/ml | ALA4766304 | ng.hr.mL-1 | ||||
| 8. | GPR40 Activator 1 | 18 | Activity | 0 | ALA4766302 | Not Active | Homo sapiens | |||||
| 9. | GPR40 Activator 1 | 18 | Activity | 0 | ALA4766301 | Not Active | Homo sapiens | |||||
| 10. | GPR40 Activator 1 | 18 | Activity | 0 | ALA4766300 | Not Active | Homo sapiens | |||||
| 11. | GPR40 Activator 1 | 18 | PPB | > | 99 | % | ALA4766299 | % | ||||
| 12. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766298 | Metabolite_Detected | ||||||
| 13. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766297 | Metabolite_Detected | ||||||
| 14. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766296 | Metabolite_Detected | ||||||
| 15. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766295 | Metabolite_Detected | ||||||
| 16. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766294 | Metabolite_Detected | ||||||
| 17. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766293 | Metabolite_Detected | ||||||
| 18. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766292 | Metabolite_Detected | ||||||
| 19. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766291 | Metabolite_Detected | ||||||
| 20. | GPR40 Activator 1 | 18 | Drug metabolism | 0 | ALA4766290 | Metabolite_Detected |
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