| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4782111 | 28f; ACT-1004-1239 | IC50 | = | 1.15 | nM | ALA4706434 | 8.94 | nM | Homo sapiens | ||
| 2. | ALA4782111 | 28f; ACT-1004-1239 | Activity | 0 | ALA4706433 | Tde | ||||||
| 3. | ALA4782111 | 28f; ACT-1004-1239 | Cp | = | 14 | ng/ml | ALA4706409 | ng/ml | ||||
| 4. | ALA4782111 | 28f; ACT-1004-1239 | Cp | = | 1.52 | ng/ml | ALA4706408 | ng/ml | ||||
| 5. | ALA4782111 | 28f; ACT-1004-1239 | Cmax | = | 4285 | ng/ml | ALA4706407 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 6. | ALA4782111 | 28f; ACT-1004-1239 | Cmax | = | 6 | ng/ml | ALA4706406 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 7. | ALA4782111 | 28f; ACT-1004-1239 | Tmax | = | 0.5 | hr | ALA4706405 | hr | ||||
| 8. | ALA4782111 | 28f; ACT-1004-1239 | Drug uptake | 0 | ALA4706404 | Dose-dependent effect | ||||||
| 9. | ALA4782111 | 28f; ACT-1004-1239 | Activity | 0 | ALA4706403 | Not Active | ||||||
| 10. | ALA4782111 | 28f; ACT-1004-1239 | Activity | 0 | ALA4706402 | Not Active | ||||||
| 11. | ALA4782111 | 28f; ACT-1004-1239 | FC | = | 2.6 | ALA4706401 | ||||||
| 12. | ALA4782111 | 28f; ACT-1004-1239 | Activity | 0 | ALA4706400 | Not Active | ||||||
| 13. | ALA4782111 | 28f; ACT-1004-1239 | FC | = | 4.9 | ALA4706399 | ||||||
| 14. | ALA4782111 | 28f; ACT-1004-1239 | FC | = | 4.1 | ALA4706398 | ||||||
| 15. | ALA4782111 | 28f; ACT-1004-1239 | Activity | 0 | ALA4706397 | Active | ||||||
| 16. | ALA4782111 | 28f; ACT-1004-1239 | IC50 | = | 0.9 | nM | ALA4706396 | 9.05 | nM | Homo sapiens | ||
| 17. | ALA4782111 | 28f; ACT-1004-1239 | IC50 | = | 0.903 | nM | ALA4706395 | 9.04 | nM | Homo sapiens | ||
| 18. | ALA4782111 | 28f; ACT-1004-1239 | IC50 | = | 0.962 | nM | ALA4706394 | 9.02 | nM | Homo sapiens | ||
| 19. | ALA4782111 | 28f; ACT-1004-1239 | IC50 | = | 0.864 | nM | ALA4706393 | 9.06 | nM | Homo sapiens | ||
| 20. | ALA4782111 | 28f; ACT-1004-1239 | IC50 | = | 0.985 | nM | ALA4706392 | 9.01 | nM | Homo sapiens |
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