| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4782157 | 78 | Ki | = | 1.5 | nM | ALA4705223 | 8.82 | nM | Homo sapiens | ||
| 2. | ALA4782157 | 78 | t1/2 | = | 113 | min | ALA4705222 | hr | ||||
| 3. | ALA4782157 | 78 | t1/2 | > | 360 | min | ALA4705221 | hr | ||||
| 4. | ALA4782157 | 78 | Stabilty | = | 100 | % | ALA4705220 | % | ||||
| 5. | ALA4782157 | 78 | Stabilty | = | 98.2 | % | ALA4705219 | % | ||||
| 6. | ALA4782157 | 78 | Stabilty | = | 100 | % | ALA4705218 | % | Sus scrofa | |||
| 7. | ALA4782157 | 78 | Stabilty | = | 2.5 | % | ALA4705217 | % | Bos taurus | |||
| 8. | ALA4782157 | 78 | PPB | = | 98.5 | % | ALA4705216 | % | ||||
| 9. | ALA4782157 | 78 | t1/2 | = | 0.66 | hr | ALA4705215 | hr | ||||
| 10. | ALA4782157 | 78 | Vdss | = | 0.23 | L/Kg | ALA4705214 | L.kg-1 | ||||
| 11. | ALA4782157 | 78 | CL | = | 16 | ml/min.kg | ALA4705213 | mL.min-1.kg-1 | ||||
| 12. | ALA4782157 | 78 | AUC | = | 839.9 | nM.hr | ALA4705212 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 13. | ALA4782157 | 78 | AUC | = | 840.94 | nM.hr | ALA4705211 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 |
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