# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4783190 | 6 | pKa | = | 7.7 | ALA4766402 | ||||||
2. | ALA4783190 | 6 | pKa | = | 3.9 | ALA4766401 | ||||||
3. | ALA4783190 | 6 | K | = | 0.087 | /min | ALA4766310 | /min | Homo sapiens | |||
4. | ALA4783190 | 6 | Activity | 0 | ALA4766302 | Not Active | Homo sapiens | |||||
5. | ALA4783190 | 6 | Activity | 0 | ALA4766301 | Not Active | Homo sapiens | |||||
6. | ALA4783190 | 6 | Activity | 0 | ALA4766300 | Not Active | Homo sapiens | |||||
7. | ALA4783190 | 6 | PPB | > | 99 | % | ALA4766299 | % | ||||
8. | ALA4783190 | 6 | ED90 | > | 100 | mg kg-1 | ALA4766284 | mg kg-1 | Mus musculus | |||
9. | ALA4783190 | 6 | Activity | 0 | ALA4766283 | Not Active | Mus musculus | |||||
10. | ALA4783190 | 6 | Time | = | 12 | min | ALA4766282 | hr | Homo sapiens | |||
11. | ALA4783190 | 6 | Kd | = | 58 | nM | ALA4766281 | 7.24 | nM | Homo sapiens | ||
12. | ALA4783190 | 6 | Emax | = | 282 | % | ALA4766280 | % | Homo sapiens | |||
13. | ALA4783190 | 6 | EC50 | = | 39 | nM | ALA4766279 | 7.41 | nM | Homo sapiens | ||
14. | ALA4783190 | 6 | Emax | = | 114 | % | ALA4766278 | % | Rattus norvegicus | |||
15. | ALA4783190 | 6 | EC50 | = | 160 | nM | ALA4766277 | 6.80 | nM | Rattus norvegicus | ||
16. | ALA4783190 | 6 | Emax | = | 127 | % | ALA4766276 | % | Mus musculus | |||
17. | ALA4783190 | 6 | EC50 | = | 32 | nM | ALA4766275 | 7.50 | nM | Mus musculus | ||
18. | ALA4783190 | 6 | Emax | = | 144 | % | ALA4766274 | % | Homo sapiens | |||
19. | ALA4783190 | 6 | EC50 | = | 340 | nM | ALA4766273 | 6.47 | nM | Homo sapiens | ||
20. | ALA4783190 | 6 | Emax | = | 80 | % | ALA4766272 | % | Homo sapiens |