# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4783492 | 19 | Activity | = | 26.3 | % | ALA4673831 | % | Homo sapiens | |||
2. | ALA4783492 | 19 | IC50 | = | 0.001 | uM | ALA4673830 | 9.05 | nM | Homo sapiens | ||
3. | ALA4783492 | 19 | logD | = | 3.3 | ALA4673828 | ||||||
4. | ALA4783492 | 19 | CLH | = | 13 | microL/min/mg | ALA4673827 | mL.min-1.g-1 | ||||
5. | ALA4783492 | 19 | Fu | = | 3.9 | % | ALA4673826 | |||||
6. | ALA4783492 | 19 | solubility | = | 15 | uM | ALA4673824 | nM | ||||
7. | ALA4783492 | 19 | F | = | 37 | % | ALA4673823 | % | ||||
8. | ALA4783492 | 19 | CL | = | 9 | ml/min.kg | ALA4673822 | mL.min-1.kg-1 | ||||
9. | ALA4783492 | 19 | Vdss | = | 0.9 | L/Kg | ALA4673821 | L.kg-1 | ||||
10. | ALA4783492 | 19 | Papp | = | 24 | 10^-6 cm/s | ALA4673820 | 10^-6 cm/s | ||||
11. | ALA4783492 | 19 | t1/2 | = | 3 | hr | ALA4673819 | hr | ||||
12. | ALA4783492 | 19 | Ratio | = | 0.5 | ALA4673818 | ||||||
13. | ALA4783492 | 19 | Kd | = | 0.001 | uM | ALA4673817 | 9.30 | nM | Homo sapiens | ||
14. | ALA4783492 | 19 | t1/2 | = | 8.7 | min | ALA4673816 | hr | Homo sapiens | |||
15. | ALA4783492 | 19 | EC50 | = | 0.007 | uM | ALA4673815 | 8.15 | nM | Homo sapiens | ||
16. | ALA4783492 | 19 | GI50 | = | 12 | uM | ALA4673814 | nM | Homo sapiens | |||
17. | ALA4783492 | 19 | GI50 | = | 13.9 | uM | ALA4673813 | nM | Homo sapiens | |||
18. | ALA4783492 | 19 | GI50 | = | 5.8 | uM | ALA4673812 | nM | Homo sapiens | |||
19. | ALA4783492 | 19 | GI50 | = | 14.4 | uM | ALA4673811 | nM | Homo sapiens | |||
20. | ALA4783492 | 19 | Activity | 0 | ALA4673810 | Not Active | Homo sapiens |