| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4783768 | IIk; C-2053 | deltaTm | = | 3.4 | degrees C | ALA4773247 | degrees C | ||||
| 2. | ALA4783768 | IIk; C-2053 | deltaTm | = | 23.7 | degrees C | ALA4773246 | degrees C | Homo sapiens | |||
| 3. | ALA4783768 | IIk; C-2053 | deltaTm | = | 23.3 | degrees C | ALA4773245 | degrees C | Homo sapiens | |||
| 4. | ALA4783768 | IIk; C-2053 | deltaTm | = | 21.9 | degrees C | ALA4773244 | degrees C | Homo sapiens | |||
| 5. | ALA4783768 | IIk; C-2053 | MTD | = | 120 | mg kg-1 | ALA4773241 | mg kg-1 | ||||
| 6. | ALA4783768 | IIk; C-2053 | MTD | = | 60 | mg kg-1 | ALA4773237 | mg kg-1 | ||||
| 7. | ALA4783768 | IIk; C-2053 | TGI | = | 62 | % | ALA4773234 | % | Homo sapiens | |||
| 8. | ALA4783768 | IIk; C-2053 | TGI | = | 47 | % | ALA4773233 | % | Homo sapiens | |||
| 9. | ALA4783768 | IIk; C-2053 | TGI | = | 84 | % | ALA4773232 | % | Homo sapiens | |||
| 10. | ALA4783768 | IIk; C-2053 | T/C | = | 350 | % | ALA4773152 | % | Rattus norvegicus | |||
| 11. | ALA4783768 | IIk; C-2053 | IC50 | = | 1.176 | uM | ALA4773139 | 5.93 | nM | Homo sapiens | ||
| 12. | ALA4783768 | IIk; C-2053 | IC50 | = | 0.224 | uM | ALA4773138 | 6.65 | nM | Homo sapiens | ||
| 13. | ALA4783768 | IIk; C-2053 | IC50 | = | 0.087 | uM | ALA4773137 | 7.06 | nM | Homo sapiens | ||
| 14. | ALA4783768 | IIk; C-2053 | IC50 | = | 0.098 | uM | ALA4773136 | 7.01 | nM | Homo sapiens | ||
| 15. | ALA4783768 | IIk; C-2053 | IC50 | = | 0.065 | uM | ALA4773132 | 7.19 | nM | Homo sapiens | ||
| 16. | ALA4783768 | IIk; C-2053 | IC50 | = | 0.025 | uM | ALA4773131 | 7.60 | nM | Homo sapiens | ||
| 17. | ALA4783768 | IIk; C-2053 | IC50 | = | 0.065 | uM | ALA4773127 | 7.19 | nM | Homo sapiens |
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