| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4785375 | 2dA; FCW66 | Papp | = | 9 | ucm/s | ALA4775623 | ucm/s | ||||
| 2. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775622 | Active | % | |||||
| 3. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775621 | Active | % | |||||
| 4. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775620 | Active | % | |||||
| 5. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775619 | Dose-dependent effect | % | |||||
| 6. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775618 | Dose-dependent effect | % | |||||
| 7. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775617 | Dose-dependent effect | % | |||||
| 8. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775616 | Dose-dependent effect | % | |||||
| 9. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775615 | Dose-dependent effect | % | |||||
| 10. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775598 | Active | % | |||||
| 11. | ALA4785375 | 2dA; FCW66 | INH | 0 | ALA4775597 | Active | % | Homo sapiens | ||||
| 12. | ALA4785375 | 2dA; FCW66 | IC50 | = | 12 | uM | ALA4775596 | 4.92 | nM | Homo sapiens | ||
| 13. | ALA4785375 | 2dA; FCW66 | Survival | > | 90 | % | ALA4775595 | % | Homo sapiens | |||
| 14. | ALA4785375 | 2dA; FCW66 | Ratio IC50 | > | 102 | ALA4775594 | ||||||
| 15. | ALA4785375 | 2dA; FCW66 | Selectivity ratio | <= | 990 | ALA4775592 | ||||||
| 16. | ALA4785375 | 2dA; FCW66 | Selectivity ratio | > | 495 | ALA4775591 | ||||||
| 17. | ALA4785375 | 2dA; FCW66 | INH | = | 50 | % | ALA4775589 | % | Rattus norvegicus | |||
| 18. | ALA4785375 | 2dA; FCW66 | INH | = | 0 | % | ALA4775588 | % | Rattus norvegicus | |||
| 19. | ALA4785375 | 2dA; FCW66 | IC50 | = | 4.9 | uM | ALA4775586 | 5.31 | nM | Homo sapiens | ||
| 20. | ALA4785375 | 2dA; FCW66 | IC50 | = | 1.01 | uM | ALA4775585 | 6.00 | nM | Rattus norvegicus |
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