# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4786439 | 16c | F | = | 70.3 | % | ALA4769715 | % | ||||
2. | ALA4786439 | 16c | AUC | = | 2059.1 | hr.ng/ml | ALA4769714 | ng.hr.mL-1 | ||||
3. | ALA4786439 | 16c | Cmax | = | 736.4 | ng/ml | ALA4769713 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
4. | ALA4786439 | 16c | t1/2 | = | 0.9 | hr | ALA4769712 | hr | ||||
5. | ALA4786439 | 16c | AUC | = | 293 | hr.ng/ml | ALA4769711 | ng.hr.mL-1 | ||||
6. | ALA4786439 | 16c | Vdss | = | 2.2 | L/Kg | ALA4769710 | L.kg-1 | ||||
7. | ALA4786439 | 16c | CL | = | 3.1 | L/hr/kg | ALA4769709 | mL.min-1.kg-1 | ||||
8. | ALA4786439 | 16c | t1/2 | = | 0.6 | hr | ALA4769708 | hr | ||||
9. | ALA4786439 | 16c | IC50 | = | 45.3 | nM | ALA4769707 | 7.34 | nM | Mus musculus | ||
10. | ALA4786439 | 16c | IC50 | = | 26 | nM | ALA4769705 | 7.58 | nM | Homo sapiens |