| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4787039 | 18a | log Ks | = | 5.3 | ALA4710765 | ||||||
| 2. | ALA4787039 | 18a | log Ks | = | 5.2 | ALA4710764 | ||||||
| 3. | ALA4787039 | 18a | log Ks | = | 5.1 | ALA4710763 | ||||||
| 4. | ALA4787039 | 18a | log Ks | = | 5.9 | ALA4710762 | Bos taurus | |||||
| 5. | ALA4787039 | 18a | Ratio IC50 | > | 530 | ALA4710761 | ||||||
| 6. | ALA4787039 | 18a | IC50 | > | 250 | uM | ALA4710760 | nM | Rattus norvegicus | |||
| 7. | ALA4787039 | 18a | IC90 | = | 1.82 | uM | ALA4710759 | nM | Trypanosoma brucei brucei | |||
| 8. | ALA4787039 | 18a | IC50 | = | 0.47 | uM | ALA4710759 | 6.33 | nM | Trypanosoma brucei brucei | ||
| 9. | ALA4787039 | 18a | INH | > | 90 | % | ALA4710758 | % | Trypanosoma brucei brucei | |||
| 10. | ALA4787039 | 18a | INH | = | 100 | % | ALA4710756 | % | Trypanosoma brucei brucei | |||
| 11. | ALA4787039 | 18a | deltaTm | = | 4.5 | degrees C | ALA4710755 | degrees C | ||||
| 12. | ALA4787039 | 18a | deltaTm | = | 6.4 | degrees C | ALA4710754 | degrees C | Bos taurus | |||
| 13. | ALA4787039 | 18a | deltaTm | = | 17.9 | degrees C | ALA4710753 | degrees C | ||||
| 14. | ALA4787039 | 18a | Activity | 0 | ALA4710752 | Active | Homo sapiens | |||||
| 15. | ALA4787039 | 18a | Activity | 0 | ALA4710751 | Active | Homo sapiens | |||||
| 16. | ALA4787039 | 18a | Papp | = | 0.27 | 10^-6 cm/s | ALA4710750 | 10^-6 cm/s | ||||
| 17. | ALA4787039 | 18a | Papp | = | 0.63 | 10^-6 cm/s | ALA4710749 | 10^-6 cm/s | ||||
| 18. | ALA4787039 | 18a | Ratio | = | 2.38 | ALA4710748 | ||||||
| 19. | ALA4787039 | 18a | Ratio IC50 | > | 2 | ALA4710746 | Trypanosoma brucei brucei |
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