# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4787753 | SBL-MC-45 | Ratio Ki | = | 6.4 | ALA4775181 | ||||||
2. | ALA4787753 | SBL-MC-45 | Ki | = | 1380 | pM | ALA4775180 | 8.86 | nM | Homo sapiens | ||
3. | ALA4787753 | SBL-MC-45 | pKi | = | 8.86 | ALA4775180 | 8.86 | nM | Homo sapiens | |||
4. | ALA4787753 | SBL-MC-45 | Ki | = | 8872 | pM | ALA4775179 | 8.05 | nM | Homo sapiens | ||
5. | ALA4787753 | SBL-MC-45 | pKi | = | 8.05 | ALA4775179 | 8.05 | nM | Homo sapiens | |||
6. | ALA4787753 | SBL-MC-45 | Selectivity Index | = | 3.33 | ALA4775178 | ||||||
7. | ALA4787753 | SBL-MC-45 | Selectivity Index | = | 0.3 | ALA4775177 | ||||||
8. | ALA4787753 | SBL-MC-45 | Efficacy | = | 101 | % | ALA4775176 | % | Homo sapiens | |||
9. | ALA4787753 | SBL-MC-45 | EC50 | = | 136 | nM | ALA4775175 | 6.87 | nM | Homo sapiens | ||
10. | ALA4787753 | SBL-MC-45 | pEC50 | = | 6.87 | ALA4775175 | 6.87 | nM | Homo sapiens | |||
11. | ALA4787753 | SBL-MC-45 | Efficacy | = | 108 | % | ALA4775174 | % | Homo sapiens | |||
12. | ALA4787753 | SBL-MC-45 | EC50 | = | 141 | nM | ALA4775173 | 6.85 | nM | Homo sapiens | ||
13. | ALA4787753 | SBL-MC-45 | pEC50 | = | 7.39 | ALA4775173 | 7.39 | nM | Homo sapiens |