# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4788651 | 6 | IC50 | > | 10 | uM | ALA4769951 | nM | Homo sapiens | |||
2. | ALA4788651 | 6 | INH | = | 97 | % | ALA4769950 | % | Homo sapiens | |||
3. | ALA4788651 | 6 | INH | = | 89.9 | % | ALA4769949 | % | Homo sapiens | |||
4. | ALA4788651 | 6 | INH | = | 60.4 | % | ALA4769948 | % | Homo sapiens | |||
5. | ALA4788651 | 6 | INH | = | 60.4 | % | ALA4769947 | % | Homo sapiens | |||
6. | ALA4788651 | 6 | INH | = | 49.5 | % | ALA4769946 | % | Homo sapiens | |||
7. | ALA4788651 | 6 | INH | < | 50 | % | ALA4769945 | % | Homo sapiens | |||
8. | ALA4788651 | 6 | INH | < | 50 | % | ALA4769944 | % | Homo sapiens | |||
9. | ALA4788651 | 6 | INH | < | 50 | % | ALA4769943 | % | Homo sapiens | |||
10. | ALA4788651 | 6 | INH | < | 50 | % | ALA4769942 | % | Homo sapiens | |||
11. | ALA4788651 | 6 | INH | < | 50 | % | ALA4769941 | % | Homo sapiens | |||
12. | ALA4788651 | 6 | t1/2 | = | 6 | min | ALA4769940 | hr | ||||
13. | ALA4788651 | 6 | t1/2 | = | 3 | min | ALA4769939 | hr | ||||
14. | ALA4788651 | 6 | permeability | = | 85.3 | 10^-6 cm/s | ALA4769938 | 10^-6 cm/s | ||||
15. | ALA4788651 | 6 | permeability | = | 10.8 | 10^-6 cm/s | ALA4769937 | 10^-6 cm/s | ||||
16. | ALA4788651 | 6 | solubility | = | 76.2 | uM | ALA4769936 | nM | ||||
17. | ALA4788651 | 6 | Fu | = | 13.8 | % | ALA4769935 | |||||
18. | ALA4788651 | 6 | Fu | = | 4.7 | % | ALA4769934 | |||||
19. | ALA4788651 | 6 | INH | = | 6 | % | ALA4769933 | % | Homo sapiens | |||
20. | ALA4788651 | 6 | INH | = | 4 | % | ALA4769932 | % | Homo sapiens |