# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BMS-986202 | 7; BMS-986202 | Ratio IC50 | = | 8 | ALA4775583 | ||||||
2. | BMS-986202 | 7; BMS-986202 | IC50 | > | 10 | uM | ALA4775582 | nM | Homo sapiens | |||
3. | BMS-986202 | 7; BMS-986202 | IC50 | > | 12.5 | uM | ALA4775581 | nM | Homo sapiens | |||
4. | BMS-986202 | 7; BMS-986202 | IC50 | = | 7.8 | nM | ALA4775580 | 8.11 | nM | Homo sapiens | ||
5. | BMS-986202 | 7; BMS-986202 | IC50 | = | 14 | uM | ALA4775579 | 4.85 | nM | Homo sapiens | ||
6. | BMS-986202 | 7; BMS-986202 | IC50 | > | 40 | uM | ALA4775578 | nM | Homo sapiens | |||
7. | BMS-986202 | 7; BMS-986202 | IC50 | > | 40 | uM | ALA4775577 | nM | Homo sapiens | |||
8. | BMS-986202 | 7; BMS-986202 | IC50 | > | 40 | uM | ALA4775576 | nM | Homo sapiens | |||
9. | BMS-986202 | 7; BMS-986202 | IC50 | > | 40 | uM | ALA4775575 | nM | Homo sapiens | |||
10. | BMS-986202 | 7; BMS-986202 | IC50 | > | 40 | uM | ALA4775574 | nM | Homo sapiens | |||
11. | BMS-986202 | 7; BMS-986202 | PB | = | 89.3 | % | ALA4775573 | % | ||||
12. | BMS-986202 | 7; BMS-986202 | PB | = | 93.3 | % | ALA4775572 | % | ||||
13. | BMS-986202 | 7; BMS-986202 | PB | = | 96 | % | ALA4775571 | % | ||||
14. | BMS-986202 | 7; BMS-986202 | PB | = | 92.4 | % | ALA4775570 | % | ||||
15. | BMS-986202 | 7; BMS-986202 | t1/2 | = | 89 | min | ALA4775569 | hr | ||||
16. | BMS-986202 | 7; BMS-986202 | t1/2 | > | 120 | min | ALA4775568 | hr | ||||
17. | BMS-986202 | 7; BMS-986202 | t1/2 | > | 120 | min | ALA4775567 | hr | ||||
18. | BMS-986202 | 7; BMS-986202 | t1/2 | > | 120 | min | ALA4775566 | hr | ||||
19. | BMS-986202 | 7; BMS-986202 | t1/2 | > | 120 | min | ALA4775565 | hr | ||||
20. | BMS-986202 | 7; BMS-986202 | IC50 | = | 481 | nM | ALA4775564 | 6.32 | nM | Mus musculus |