# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4790634 | 9x | TGI | > | 60 | % | ALA4710046 | % | Mus musculus | |||
2. | ALA4790634 | 9x | TGI | > | 60 | % | ALA4710045 | % | Mus musculus | |||
3. | ALA4790634 | 9x | Activity | 0 | ALA4710044 | Non-Toxic | ||||||
4. | ALA4790634 | 9x | Activity | 0 | ALA4710043 | Non-Toxic | ||||||
5. | ALA4790634 | 9x | Activity | 0 | ALA4710042 | Active | Mus musculus | |||||
6. | ALA4790634 | 9x | Activity | 0 | ALA4710041 | Active | Mus musculus | |||||
7. | ALA4790634 | 9x | Activity | 0 | ALA4710040 | Active | Mus musculus | |||||
8. | ALA4790634 | 9x | Activity | 0 | ALA4710039 | Active | Mus musculus | |||||
9. | ALA4790634 | 9x | INH | 0 | ALA4710038 | Dose-dependent effect | % | |||||
10. | ALA4790634 | 9x | INH | 0 | ALA4710037 | Dose-dependent effect | % | |||||
11. | ALA4790634 | 9x | INH | 0 | ALA4710036 | Dose-dependent effect | % | |||||
12. | ALA4790634 | 9x | INH | 0 | ALA4710035 | Dose-dependent effect | % | |||||
13. | ALA4790634 | 9x | Activity | 0 | ALA4710034 | Dose-dependent effect | Mus musculus | |||||
14. | ALA4790634 | 9x | Activity | 0 | ALA4710033 | Dose-dependent effect | Mus musculus | |||||
15. | ALA4790634 | 9x | F | = | 3 | % | ALA4710032 | % | ||||
16. | ALA4790634 | 9x | AUC | = | 2343 | ng.hr/ml | ALA4710031 | ng.hr.mL-1 | ||||
17. | ALA4790634 | 9x | AUCt | = | 2112 | ng.hr/ml | ALA4710030 | ng.hr.mL-1 | ||||
18. | ALA4790634 | 9x | Cmax | = | 194 | ng/ml | ALA4710029 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
19. | ALA4790634 | 9x | Tmax | = | 0.75 | hr | ALA4710028 | hr | ||||
20. | ALA4790634 | 9x | t1/2 | = | 7.59 | hr | ALA4710027 | hr |