# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4790764 | 75 | PPB | = | 97.5 | % | ALA4705237 | % | ||||
2. | ALA4790764 | 75 | t1/2 | = | 2.84 | hr | ALA4705236 | hr | ||||
3. | ALA4790764 | 75 | Vdss | = | 1.06 | L/Kg | ALA4705235 | L.kg-1 | ||||
4. | ALA4790764 | 75 | CL | = | 20.15 | ml/min.kg | ALA4705234 | mL.min-1.kg-1 | ||||
5. | ALA4790764 | 75 | AUC | = | 303.71 | nM.hr | ALA4705233 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
6. | ALA4790764 | 75 | AUC | = | 306.1 | nM.hr | ALA4705232 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
7. | ALA4790764 | 75 | PPB | = | 99.7 | % | ALA4705231 | % | ||||
8. | ALA4790764 | 75 | t1/2 | = | 0.06 | hr | ALA4705230 | hr | ||||
9. | ALA4790764 | 75 | Vdss | = | 0.48 | L/Kg | ALA4705229 | L.kg-1 | ||||
10. | ALA4790764 | 75 | CL | = | 107 | ml/min.kg | ALA4705228 | mL.min-1.kg-1 | ||||
11. | ALA4790764 | 75 | AUC | = | 19.4 | nM.hr | ALA4705227 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
12. | ALA4790764 | 75 | AUC | = | 23.3 | nM.hr | ALA4705226 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
13. | ALA4790764 | 75 | Ki | = | 1.36 | nM | ALA4705223 | 8.87 | nM | Homo sapiens | ||
14. | ALA4790764 | 75 | t1/2 | > | 360 | min | ALA4705222 | hr | ||||
15. | ALA4790764 | 75 | t1/2 | 0 | ALA4705221 | Not Determined | ||||||
16. | ALA4790764 | 75 | Stabilty | = | 99.2 | % | ALA4705220 | % | ||||
17. | ALA4790764 | 75 | Stabilty | = | 98.9 | % | ALA4705219 | % | ||||
18. | ALA4790764 | 75 | Stabilty | = | 96.6 | % | ALA4705218 | % | Sus scrofa | |||
19. | ALA4790764 | 75 | Stabilty | = | 91.8 | % | ALA4705217 | % | Bos taurus | |||
20. | ALA4790764 | 75 | Ki | = | 1.36 | nM | ALA5035794 | 8.87 | nM | Homo sapiens |