# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4791246 | 5; IPR-3242 | Activity | = | 17 | % | ALA4679634 | % | ||||
2. | ALA4791246 | 5; IPR-3242 | %max | = | 47 | % | ALA4679633 | % | Homo sapiens | |||
3. | ALA4791246 | 5; IPR-3242 | Activity | 0 | ALA4679632 | Not Active | ||||||
4. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679631 | Not Active | % | Homo sapiens | ||||
5. | ALA4791246 | 5; IPR-3242 | Activity | 0 | ALA4679630 | Not Active | Homo sapiens | |||||
6. | ALA4791246 | 5; IPR-3242 | IC50 | = | 4.9 | uM | ALA4679629 | 5.31 | nM | Homo sapiens | ||
7. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679629 | Dose-dependent effect | % | Homo sapiens | ||||
8. | ALA4791246 | 5; IPR-3242 | IC50 | = | 0.5 | uM | ALA4679628 | 6.30 | nM | Homo sapiens | ||
9. | ALA4791246 | 5; IPR-3242 | IC50 | = | 8.6 | uM | ALA4679627 | 5.07 | nM | Homo sapiens | ||
10. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679627 | Dose-dependent effect | % | Homo sapiens | ||||
11. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679626 | Not Active | % | Homo sapiens | ||||
12. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679625 | Not Active | % | Homo sapiens | ||||
13. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679624 | Not Active | % | Homo sapiens | ||||
14. | ALA4791246 | 5; IPR-3242 | Drug metabolism | 0 | ALA4679623 | Metabolite_Notdetected | ||||||
15. | ALA4791246 | 5; IPR-3242 | INH | 0 | ALA4679622 | Active | % | Homo sapiens | ||||
16. | ALA4791246 | 5; IPR-3242 | Activity | = | 150 | nm | ALA4679621 | nm |