# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4791842 | 24 | pKa | = | 8.6 | ALA4766402 | ||||||
2. | ALA4791842 | 24 | pKa | = | 4.6 | ALA4766401 | ||||||
3. | ALA4791842 | 24 | Activity | 0 | ALA4766302 | Not Active | Homo sapiens | |||||
4. | ALA4791842 | 24 | Activity | 0 | ALA4766301 | Not Active | Homo sapiens | |||||
5. | ALA4791842 | 24 | Activity | 0 | ALA4766300 | Not Active | Homo sapiens | |||||
6. | ALA4791842 | 24 | PPB | > | 99 | % | ALA4766299 | % | ||||
7. | ALA4791842 | 24 | ED90 | = | 22 | mg kg-1 | ALA4766284 | mg kg-1 | Mus musculus | |||
8. | ALA4791842 | 24 | Activity | 0 | ALA4766283 | Active | Mus musculus | |||||
9. | ALA4791842 | 24 | Time | = | 66 | min | ALA4766282 | hr | Homo sapiens | |||
10. | ALA4791842 | 24 | Kd | = | 2.2 | nM | ALA4766281 | 8.66 | nM | Homo sapiens | ||
11. | ALA4791842 | 24 | Emax | = | 249 | % | ALA4766280 | % | Homo sapiens | |||
12. | ALA4791842 | 24 | EC50 | = | 6.2 | nM | ALA4766279 | 8.21 | nM | Homo sapiens | ||
13. | ALA4791842 | 24 | Emax | = | 135 | % | ALA4766278 | % | Rattus norvegicus | |||
14. | ALA4791842 | 24 | EC50 | = | 1.3 | nM | ALA4766277 | 8.89 | nM | Rattus norvegicus | ||
15. | ALA4791842 | 24 | Emax | = | 135 | % | ALA4766276 | % | Mus musculus | |||
16. | ALA4791842 | 24 | EC50 | = | 0.88 | nM | ALA4766275 | 9.06 | nM | Mus musculus | ||
17. | ALA4791842 | 24 | Emax | = | 137 | % | ALA4766274 | % | Homo sapiens | |||
18. | ALA4791842 | 24 | EC50 | = | 11 | nM | ALA4766273 | 7.96 | nM | Homo sapiens | ||
19. | ALA4791842 | 24 | Emax | = | 46 | % | ALA4766272 | % | Homo sapiens | |||
20. | ALA4791842 | 24 | EC50 | = | 19 | nM | ALA4766271 | 7.72 | nM | Homo sapiens |