# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4793665 | 47 | IC50 | = | 0.017 | uM | ALA4674513 | 7.77 | nM | Homo sapiens | ||
2. | ALA4793665 | 47 | IC50 | = | 0.078 | uM | ALA4674512 | 7.11 | nM | Homo sapiens | ||
3. | ALA4793665 | 47 | IC50 | = | 0.711 | uM | ALA4674511 | 6.15 | nM | Homo sapiens | ||
4. | ALA4793665 | 47 | Papp | = | 13.4 | 10^-6 cm/s | ALA4674509 | 10^-6 cm/s | ||||
5. | ALA4793665 | 47 | Fu | = | 16 | % | ALA4674508 | |||||
6. | ALA4793665 | 47 | Ratio | = | 1.1 | ALA4674507 | ||||||
7. | ALA4793665 | 47 | AUC | = | 31.9 | ng/mL.hr | ALA4674506 | ng.hr.mL-1 | ||||
8. | ALA4793665 | 47 | CL | = | 54.7 | ml/min.kg | ALA4674505 | mL.min-1.kg-1 | ||||
9. | ALA4793665 | 47 | t1/2 | = | 0.7 | hr | ALA4674504 | hr | ||||
10. | ALA4793665 | 47 | IC50 | = | 8.6 | nM | ALA4674072 | 8.07 | nM | Homo sapiens | ||
11. | ALA4793665 | 47 | IC50 | = | 10.2 | nM | ALA4674071 | 7.99 | nM | Homo sapiens | ||
12. | ALA4793665 | 47 | IC50 | = | 0.09 | nM | ALA4674070 | 10.05 | nM | Homo sapiens | ||
13. | ALA4793665 | 47 | IC50 | = | 6.4 | nM | ALA4674069 | 8.19 | nM | Homo sapiens |