| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4794465 | 3 | Fu | = | 0.1 | % | ALA4700787 | |||||
| 2. | ALA4794465 | 3 | logD | = | 4.42 | ALA4700786 | ||||||
| 3. | ALA4794465 | 3 | Activity | 0 | ALA4700780 | Toxic | ||||||
| 4. | ALA4794465 | 3 | IC50 | = | 690 | nM | ALA4700779 | 6.16 | nM | Homo sapiens | ||
| 5. | ALA4794465 | 3 | IC50 | = | 1.4 | uM | ALA4700778 | 5.85 | nM | Homo sapiens | ||
| 6. | ALA4794465 | 3 | Activity | 0 | ALA4700777 | Toxic | ||||||
| 7. | ALA4794465 | 3 | NOAEL | = | 15 | uM | ALA4700776 | uM | ||||
| 8. | ALA4794465 | 3 | IC50 | = | 200 | nM | ALA4700775 | 6.70 | nM | Homo sapiens | ||
| 9. | ALA4794465 | 3 | F | = | 44 | % | ALA4700774 | % | ||||
| 10. | ALA4794465 | 3 | F | = | 64 | % | ALA4700773 | % | ||||
| 11. | ALA4794465 | 3 | F | = | 49 | % | ALA4700772 | % | ||||
| 12. | ALA4794465 | 3 | Activity | = | 25 | % | ALA4700771 | % | Canis lupus familiaris | |||
| 13. | ALA4794465 | 3 | Activity | = | 25 | % | ALA4700770 | % | Macaca fascicularis | |||
| 14. | ALA4794465 | 3 | Activity | = | 25 | % | ALA4700769 | % | Rattus norvegicus | |||
| 15. | ALA4794465 | 3 | AUC | = | 7.6 | uM.hr | ALA4700768 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 16. | ALA4794465 | 3 | Stabilty | = | 96 | % | ALA4700767 | % | ||||
| 17. | ALA4794465 | 3 | Cp | = | 1.7 | uM | ALA4700766 | uM | ||||
| 18. | ALA4794465 | 3 | Cp | = | 2.1 | uM | ALA4700765 | uM | ||||
| 19. | ALA4794465 | 3 | INH | = | 59 | % | ALA4700764 | % | ||||
| 20. | ALA4794465 | 3 | BPR | = | 0.38 | ALA4700763 |
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