| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4794972 | 1 | IC50 | = | 0.3 | uM | ALA5217199 | 6.52 | nM | Rattus norvegicus | ||
| 2. | ALA4794972 | 1 | t1/2 | = | 3 | hr | ALA5217197 | hr | ||||
| 3. | ALA4794972 | 1 | Tmax | = | 2.7 | hr | ALA5217195 | hr | ||||
| 4. | ALA4794972 | 1 | fCmax | < | 43 | nM | ALA5217193 | nM | ||||
| 5. | ALA4794972 | 1 | Cmax | = | 6120 | nM | ALA5217191 | nM | ||||
| 6. | ALA4794972 | 1 | AUC | = | 37100 | nM.hr | ALA5217189 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 7. | ALA4794972 | 1 | F | = | 50 | % | ALA5217188 | % | ||||
| 8. | ALA4794972 | 1 | t1/2 | = | 5.2 | hr | ALA5217187 | hr | ||||
| 9. | ALA4794972 | 1 | t1/2 | = | 2 | hr | ALA5217186 | hr | ||||
| 10. | ALA4794972 | 1 | CL | = | 34.9 | ml/min.kg | ALA5217185 | mL.min-1.kg-1 | ||||
| 11. | ALA4794972 | 1 | Vdss | = | 3.4 | L/Kg | ALA5217184 | L.kg-1 | ||||
| 12. | ALA4794972 | 1 | fCmax | < | 30 | nM | ALA5217183 | nM | ||||
| 13. | ALA4794972 | 1 | fCmax | < | 6 | nM | ALA5217182 | nM | ||||
| 14. | ALA4794972 | 1 | Cmax | = | 4940 | nM | ALA5217181 | nM | ||||
| 15. | ALA4794972 | 1 | Cmax | = | 1020 | nM | ALA5217180 | nM | ||||
| 16. | ALA4794972 | 1 | AUC | = | 2090 | nM.hr | ALA5217179 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 17. | ALA4794972 | 1 | AUC | = | 5240 | nM.hr | ALA5217178 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 18. | ALA4794972 | 1 | Papp | = | 5.5 | nm/s | ALA5217177 | nm/s | ||||
| 19. | ALA4794972 | 1 | Fu | < | 0.006 | ALA5217176 | ||||||
| 20. | ALA4794972 | 1 | Stability | = | 59 | % | ALA5217175 | % |
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