| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  VU2957 | 9 | MED | = | 1 | mg kg-1 | ALA4665938 | mg kg-1 | Rattus norvegicus | |||
| 2. | VU2957 | 9 | IC50 | = | 12.5 | uM | ALA4665937 | 4.90 | nM | Homo sapiens | ||
| 3. | VU2957 | 9 | Emax | = | 123 | % | ALA4665936 | % | Rattus norvegicus | |||
| 4. | VU2957 | 9 | pEC50 | = | 6.71 | ALA4665935 | 6.71 | nM | Rattus norvegicus | |||
| 5. | VU2957 | 9 | EC50 | = | 197 | nM | ALA4665935 | 6.71 | nM | Rattus norvegicus | ||
| 6. | VU2957 | 9 | Kp | = | 1.5 | ALA4665934 | ||||||
| 7. | VU2957 | 9 | Activity | = | 50 | % | ALA4665933 | % | Rattus norvegicus | |||
| 8. | VU2957 | 9 | Activity | = | 93 | % | ALA4665921 | % | Homo sapiens | |||
| 9. | VU2957 | 9 | EC50 | = | 65 | nM | ALA4665920 | 7.19 | nM | Homo sapiens | ||
| 10. | VU2957 | 9 | EC50 | = | 64.6 | nM | ALA5258238 | 7.19 | nM | Homo sapiens | ||
| 11. | VU2957 | 9 | pEC50 | = | 7.19 | ALA5258238 | 7.19 | nM | Homo sapiens | |||
| 12. | VU2957 | 9 | Emax | = | 92.6 | % | ALA5258237 | % | Homo sapiens | |||
| 13. | VU2957 | 9 | pEC50 | = | 6.71 | ALA5258236 | 6.71 | nM | Rattus norvegicus | |||
| 14. | VU2957 | 9 | EC50 | = | 197 | nM | ALA5258236 | 6.71 | nM | Rattus norvegicus | ||
| 15. | VU2957 | 9 | Emax | = | 132 | % | ALA5258235 | % | Rattus norvegicus | |||
| 16. | VU2957 | 9 | EC50 | > | 10 | uM | ALA5258234 | nM | Rattus norvegicus | |||
| 17. | VU2957 | 9 | EC50 | > | 10 | uM | ALA5258233 | nM | Rattus norvegicus | |||
| 18. | VU2957 | 9 | EC50 | > | 10 | uM | ALA5258232 | nM | Rattus norvegicus | |||
| 19. | VU2957 | 9 | EC50 | > | 10 | uM | ALA5258231 | nM | Rattus norvegicus | |||
| 20. | VU2957 | 9 | EC50 | > | 10 | uM | ALA5258230 | nM | Homo sapiens |
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