# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4797826 | IIe; C-2041 | Activity | 0 | ALA4773254 | Non-Toxic | ||||||
2. | ALA4797826 | IIe; C-2041 | deltaTm | = | 5.4 | degrees C | ALA4773247 | degrees C | ||||
3. | ALA4797826 | IIe; C-2041 | deltaTm | = | 27.6 | degrees C | ALA4773246 | degrees C | Homo sapiens | |||
4. | ALA4797826 | IIe; C-2041 | deltaTm | = | 30 | degrees C | ALA4773245 | degrees C | Homo sapiens | |||
5. | ALA4797826 | IIe; C-2041 | deltaTm | = | 23.3 | degrees C | ALA4773244 | degrees C | Homo sapiens | |||
6. | ALA4797826 | IIe; C-2041 | Activity | 0 | ALA4773243 | Non-Toxic | ||||||
7. | ALA4797826 | IIe; C-2041 | Survival | = | 71 | day | ALA4773242 | day | ||||
8. | ALA4797826 | IIe; C-2041 | MTD | = | 6 | mg kg-1 | ALA4773241 | mg kg-1 | ||||
9. | ALA4797826 | IIe; C-2041 | MTD | = | 5 | mg kg-1 | ALA4773237 | mg kg-1 | ||||
10. | ALA4797826 | IIe; C-2041 | TGI | = | 53 | % | ALA4773215 | % | Homo sapiens | |||
11. | ALA4797826 | IIe; C-2041 | TGI | = | 61 | % | ALA4773214 | % | Homo sapiens | |||
12. | ALA4797826 | IIe; C-2041 | TGI | = | 29 | % | ALA4773213 | % | Homo sapiens | |||
13. | ALA4797826 | IIe; C-2041 | TGI | = | 48 | % | ALA4773212 | % | Homo sapiens | |||
14. | ALA4797826 | IIe; C-2041 | TGI | = | 81 | % | ALA4773211 | % | Homo sapiens | |||
15. | ALA4797826 | IIe; C-2041 | TGI | = | 38 | % | ALA4773210 | % | Homo sapiens | |||
16. | ALA4797826 | IIe; C-2041 | TGI | = | 80 | % | ALA4773209 | % | Homo sapiens | |||
17. | ALA4797826 | IIe; C-2041 | T/C | = | 300 | % | ALA4773150 | % | Rattus norvegicus | |||
18. | ALA4797826 | IIe; C-2041 | IC50 | = | 0.032 | uM | ALA4773140 | 7.50 | nM | Homo sapiens | ||
19. | ALA4797826 | IIe; C-2041 | IC50 | = | 0.069 | uM | ALA4773139 | 7.16 | nM | Homo sapiens | ||
20. | ALA4797826 | IIe; C-2041 | IC50 | = | 0.054 | uM | ALA4773138 | 7.27 | nM | Homo sapiens |