| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4797980 | 1e | Ratio Ki | = | 49 | ALA4770554 | ||||||
| 2. | ALA4797980 | 1e | Activity | = | 90.7 | % | ALA4770550 | % | Mus musculus | |||
| 3. | ALA4797980 | 1e | INH | 0 | ALA4770549 | Active | % | Homo sapiens | ||||
| 4. | ALA4797980 | 1e | IC50 | = | 1.907 | uM | ALA4770548 | 5.72 | nM | Homo sapiens | ||
| 5. | ALA4797980 | 1e | EC50 | = | 13.4 | uM | ALA4770547 | 4.87 | nM | Homo sapiens | ||
| 6. | ALA4797980 | 1e | EC50 | > | 100 | uM | ALA4770546 | nM | Homo sapiens | |||
| 7. | ALA4797980 | 1e | EC50 | > | 100 | uM | ALA4770545 | nM | Homo sapiens | |||
| 8. | ALA4797980 | 1e | PB | = | 99.9 | % | ALA4770544 | % | Homo sapiens | |||
| 9. | ALA4797980 | 1e | t1/2 | = | 165 | min | ALA4770543 | hr | ||||
| 10. | ALA4797980 | 1e | CLH | = | 11.5 | microL/min/mg | ALA4770542 | mL.min-1.g-1 | ||||
| 11. | ALA4797980 | 1e | t1/2 | = | 60 | min | ALA4770541 | hr | ||||
| 12. | ALA4797980 | 1e | Ki | = | 1270 | nM | ALA4770540 | 5.90 | nM | Homo sapiens | ||
| 13. | ALA4797980 | 1e | Ki | = | 25.7 | nM | ALA4770539 | 7.59 | nM | Homo sapiens | ||
| 14. | ALA4797980 | 1e | Stabilty | = | 48 | % | ALA4770538 | % |
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