# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4798141 | 12d | Ratio IC50 | = | 20 | ALA4716887 | ||||||
2. | ALA4798141 | 12d | IC50 | = | 1 | uM | ALA4716871 | 6.00 | nM | Homo sapiens | ||
3. | ALA4798141 | 12d | permeability | = | 3.1 | cm/s | ALA4716869 | cm/s | ||||
4. | ALA4798141 | 12d | permeability | = | 2.6 | cm/s | ALA4716868 | cm/s | ||||
5. | ALA4798141 | 12d | log(permeability) | = | -4.1 | ALA4716867 | ||||||
6. | ALA4798141 | 12d | solubility | > | 175 | uM | ALA4716866 | nM | ||||
7. | ALA4798141 | 12d | IC50 | = | 3.3 | uM | ALA4716865 | 5.48 | nM | Homo sapiens | ||
8. | ALA4798141 | 12d | CLH | = | 32 | microL/min/mg | ALA4716864 | mL.min-1.g-1 | ||||
9. | ALA4798141 | 12d | CLH | = | 30 | microL/min/mg | ALA4716863 | mL.min-1.g-1 | ||||
10. | ALA4798141 | 12d | CLH | = | 37 | microL/min/mg | ALA4716862 | mL.min-1.g-1 | ||||
11. | ALA4798141 | 12d | IC50 | = | 5120 | nM | ALA4716833 | 5.29 | nM | Mus musculus | ||
12. | ALA4798141 | 12d | IC50 | = | 703 | nM | ALA4716832 | 6.15 | nM | Homo sapiens | ||
13. | ALA4798141 | 12d | IC50 | = | 13 | nM | ALA4716830 | 7.89 | nM | Homo sapiens |