# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4799274 | 7g | Activity | 0 | ALA4770553 | Not Active | Mus musculus | |||||
2. | ALA4799274 | 7g | Activity | 0 | ALA4770552 | Not Active | Mus musculus | |||||
3. | ALA4799274 | 7g | Activity | 0 | ALA4770551 | Active | ||||||
4. | ALA4799274 | 7g | Activity | = | 107 | % | ALA4770550 | % | Mus musculus | |||
5. | ALA4799274 | 7g | INH | 0 | ALA4770549 | Active | % | Homo sapiens | ||||
6. | ALA4799274 | 7g | IC50 | = | 0.448 | uM | ALA4770548 | 6.35 | nM | Homo sapiens | ||
7. | ALA4799274 | 7g | EC50 | = | 14.8 | uM | ALA4770547 | 4.83 | nM | Homo sapiens | ||
8. | ALA4799274 | 7g | EC50 | = | 21.7 | uM | ALA4770546 | 4.66 | nM | Homo sapiens | ||
9. | ALA4799274 | 7g | EC50 | = | 24.7 | uM | ALA4770545 | 4.61 | nM | Homo sapiens | ||
10. | ALA4799274 | 7g | PB | = | 98.8 | % | ALA4770544 | % | Homo sapiens | |||
11. | ALA4799274 | 7g | t1/2 | = | 288 | min | ALA4770543 | hr | ||||
12. | ALA4799274 | 7g | CLH | = | 11 | microL/min/mg | ALA4770542 | mL.min-1.g-1 | ||||
13. | ALA4799274 | 7g | t1/2 | = | 63 | min | ALA4770541 | hr | ||||
14. | ALA4799274 | 7g | Ki | = | 127 | nM | ALA4770540 | 6.90 | nM | Homo sapiens | ||
15. | ALA4799274 | 7g | Ki | = | 14.7 | nM | ALA4770539 | 7.83 | nM | Homo sapiens | ||
16. | ALA4799274 | 7g | Stabilty | = | 49 | % | ALA4770538 | % |