# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4800124 | 9b | Activity | 0 | ALA4686487 | Non-Toxic | ||||||
2. | ALA4800124 | 9b | Activity | 0 | ALA4686486 | Non-Toxic | ||||||
3. | ALA4800124 | 9b | Activity | 0 | ALA4686481 | Non-Toxic | ||||||
4. | ALA4800124 | 9b | Activity | 0 | ALA4686480 | Non-Toxic | ||||||
5. | ALA4800124 | 9b | Activity | = | 4.6 | % | ALA4686475 | % | ||||
6. | ALA4800124 | 9b | Activity | = | 8.5 | % | ALA4686474 | % | ||||
7. | ALA4800124 | 9b | Activity | = | 5.7 | % | ALA4686473 | % | ||||
8. | ALA4800124 | 9b | TGI | = | 30.5 | % | ALA4686470 | % | Homo sapiens | |||
9. | ALA4800124 | 9b | TGI | = | 46.3 | % | ALA4686468 | % | Homo sapiens | |||
10. | ALA4800124 | 9b | TGI | = | 35.2 | % | ALA4686465 | % | Homo sapiens | |||
11. | ALA4800124 | 9b | TGI | 0 | ALA4686463 | Dose-dependent effect | Homo sapiens | |||||
12. | ALA4800124 | 9b | Drug metabolism | = | 98.7 | % | ALA4686462 | % | Homo sapiens | |||
13. | ALA4800124 | 9b | Drug metabolism | = | 88.7 | % | ALA4686460 | % | Homo sapiens | |||
14. | ALA4800124 | 9b | t1/2 | = | 43.8 | hr | ALA4686458 | hr | ||||
15. | ALA4800124 | 9b | t1/2 | > | 72 | hr | ALA4686457 | hr | ||||
16. | ALA4800124 | 9b | IC50 | = | 86.79 | uM | ALA4686455 | 4.06 | nM | Homo sapiens | ||
17. | ALA4800124 | 9b | IC50 | > | 200 | uM | ALA4686454 | nM | Homo sapiens | |||
18. | ALA4800124 | 9b | IC50 | = | 2.8 | 10^-3microM | ALA4686453 | 8.55 | nM | Homo sapiens | ||
19. | ALA4800124 | 9b | IC50 | = | 6.59 | uM | ALA4686452 | 5.18 | nM | Homo sapiens |