| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Denbufylline | 2 | Protection | < | 49 | % | ALA800813 | % | Rattus norvegicus | |||
| 2. | Denbufylline | 2 | IC50 | = | 0.17 | nM | ALA757135 | 9.77 | nM | Homo sapiens | ||
| 3. | Denbufylline | 2 | Rolipram activity | = | 100 | % | ALA757137 | % | Homo sapiens | |||
| 4. | Denbufylline | 2 | CTS | = | 3.5 | ALA693335 | Homo sapiens | |||||
| 5. | Denbufylline | 2 | TAR | = | 2.1 | ALA696757 | Homo sapiens | |||||
| 6. | Denbufylline | 2 | Ki | = | 31.5 | uM | ALA641988 | 4.50 | nM | Homo sapiens | ||
| 7. | Denbufylline | 2 | Ki | = | 16.5 | uM | ALA640348 | 4.78 | nM | Cavia porcellus | ||
| 8. | Denbufylline | 2 | Selectivity | = | 15.3 | ALA840643 | ||||||
| 9. | Denbufylline | 2 | Ki | = | 44.9 | uM | ALA824110 | 4.35 | nM | Homo sapiens | ||
| 10. | Denbufylline | 2 | ED15 | = | 90 | mg kg-1 | ALA823443 | mg kg-1 | Cavia porcellus | |||
| 11. | Denbufylline | 2 | ED50 | = | 5.9 | mg kg-1 | ALA822017 | mg.kg-1 | Cavia porcellus | |||
| 12. | Denbufylline | 2 | Selectivity | = | 600 | ALA849589 | ||||||
| 13. | Denbufylline | 2 | EC15 | = | 6 | uM | ALA686050 | uM | Cavia porcellus | |||
| 14. | Denbufylline | 2 | EC50 | = | 0.01 | uM | ALA685182 | 8.00 | nM | Cavia porcellus | ||
| 15. | Denbufylline | 2 | IC50 | = | 0.17 | uM | ALA765683 | nM | Homo sapiens | |||
| 16. | Denbufylline | 2 | Activity | = | 100 | % | ALA768606 | % | Homo sapiens | |||
| 17. | Denbufylline | 2 | CTS increase | = | 3.5 | ALA696913 | ||||||
| 18. | Denbufylline | 2 | CT-luci TAR | = | 2.1 | T/C | ALA653481 | T/C | ||||
| 19. | Denbufylline | 2 | Emesis | = | 3 | ALA810425 | Suncus murinus |
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