# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4845890 | 19h | INH | > | 70 | % | ALA4841129 | % | Rattus norvegicus | |||
2. | ALA4845890 | 19h | INH | = | 90 | % | ALA4841128 | % | Rattus norvegicus | |||
3. | ALA4845890 | 19h | CL | = | 0.55 | L/hr/kg | ALA4841126 | mL.min-1.kg-1 | ||||
4. | ALA4845890 | 19h | AUC | = | 26786.92 | ug/L.hr | ALA4841124 | ng.hr.mL-1 | ||||
5. | ALA4845890 | 19h | Cmax | = | 3192.06 | ug/L | ALA4841122 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
6. | ALA4845890 | 19h | Tmax | = | 0.38 | hr | ALA4841120 | hr | ||||
7. | ALA4845890 | 19h | IC50 | = | 1.1 | nM | ALA4841116 | 8.96 | nM | Homo sapiens | ||
8. | ALA4845890 | 19h | IC50 | > | 100 | nM | ALA4841115 | nM | Homo sapiens | |||
9. | ALA4845890 | 19h | Activity | > | 95 | % | ALA4841114 | % | Homo sapiens | |||
10. | ALA4845890 | 19h | IC50 | > | 100 | nM | ALA4841113 | nM | Homo sapiens | |||
11. | ALA4845890 | 19h | Stability | = | 64.07 | % | ALA4841110 | % | ||||
12. | ALA4845890 | 19h | Stability | = | 34.44 | % | ALA4841109 | % | ||||
13. | ALA4845890 | 19h | t1/2 | = | 2.43 | hr | ALA4841107 | hr |