| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4846384 | 44 | F | = | 10.4 | % | ALA4845023 | % | ||||
| 2. | ALA4846384 | 44 | AUCt/dose | = | 164 | ng/mL.hr | ALA4845022 | ng/mL.hr | ||||
| 3. | ALA4846384 | 44 | Tmax | = | 3.2 | hr | ALA4845021 | hr | ||||
| 4. | ALA4846384 | 44 | Cmax/dose | = | 21 | ng/ml | ALA4845020 | ng/ml | ||||
| 5. | ALA4846384 | 44 | t1/2 | = | 2.4 | hr | ALA4845019 | hr | ||||
| 6. | ALA4846384 | 44 | AUCt/dose | = | 1578 | ng/mL.hr | ALA4845018 | ng/mL.hr | ||||
| 7. | ALA4846384 | 44 | Vdss | = | 1.5 | L/Kg | ALA4845017 | L.kg-1 | ||||
| 8. | ALA4846384 | 44 | CL | = | 5.6 | ml/min.Kg | ALA4845016 | mL.min-1.kg-1 | ||||
| 9. | ALA4846384 | 44 | t1/2 | = | 10.5 | hr | ALA4845015 | hr | ||||
| 10. | ALA4846384 | 44 | EC50 | = | 68 | nM | ALA4845014 | 7.17 | nM | Mus musculus | ||
| 11. | ALA4846384 | 44 | EC50 | = | 38 | nM | ALA4845013 | 7.42 | nM | Mus musculus | ||
| 12. | ALA4846384 | 44 | INH | = | 9 | % | ALA4845010 | % | Homo sapiens | |||
| 13. | ALA4846384 | 44 | INH | = | 4 | % | ALA4845009 | % | Homo sapiens | |||
| 14. | ALA4846384 | 44 | IC50 | = | 11 | nM | ALA4845008 | 7.96 | nM | Homo sapiens |
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