| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4847762 | 14f | Cmax | = | 3.82 | ug/L | ALA4841375 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 2. | ALA4847762 | 14f | Vdss | = | 1.28 | L/Kg | ALA4841374 | L.kg-1 | ||||
| 3. | ALA4847762 | 14f | t1/2 | = | 0.92 | hr | ALA4841373 | hr | ||||
| 4. | ALA4847762 | 14f | CL | = | 4.05 | L/hr/kg | ALA4841372 | mL.min-1.kg-1 | ||||
| 5. | ALA4847762 | 14f | Activity | 0 | ALA4841371 | Non-Toxic | ||||||
| 6. | ALA4847762 | 14f | Activity | 0 | ALA4841370 | Non-Toxic | ||||||
| 7. | ALA4847762 | 14f | Activity | 0 | ALA4841369 | Non-Toxic | ||||||
| 8. | ALA4847762 | 14f | Activity | 0 | ALA4841368 | Non-Toxic | ||||||
| 9. | ALA4847762 | 14f | Activity | 0 | ALA4841367 | Non-Toxic | ||||||
| 10. | ALA4847762 | 14f | Activity | 0 | ALA4841366 | Non-Toxic | ||||||
| 11. | ALA4847762 | 14f | INH | 0 | ALA4841365 | Not Active | % | |||||
| 12. | ALA4847762 | 14f | INH | 0 | ALA4841364 | Not Active | % | |||||
| 13. | ALA4847762 | 14f | TGI | = | 48.7 | % | ALA4841363 | % | Homo sapiens | |||
| 14. | ALA4847762 | 14f | TGI | = | 73.4 | % | ALA4841362 | % | Homo sapiens | |||
| 15. | ALA4847762 | 14f | Ratio IC50 | = | 8 | ALA4841361 | Homo sapiens | |||||
| 16. | ALA4847762 | 14f | INH | 0 | ALA4841360 | Dose-Dependent Effect | % | Homo sapiens | ||||
| 17. | ALA4847762 | 14f | IC50 | = | 0.57 | uM | ALA4841360 | 6.24 | nM | Homo sapiens | ||
| 18. | ALA4847762 | 14f | Ratio IC50 | = | 2 | ALA4841359 | Homo sapiens | |||||
| 19. | ALA4847762 | 14f | IC50 | = | 0.983 | uM | ALA4841358 | 6.01 | nM | Homo sapiens | ||
| 20. | ALA4847762 | 14f | INH | > | 90 | % | ALA4841357 | % | Homo sapiens |
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