| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4848002 | 27; CYR715 | Activity | = | 1 | % | ALA4815929 | % | ||||
| 2. | ALA4848002 | 27; CYR715 | Activity | = | 25 | mmHg | ALA4815927 | mmHg | ||||
| 3. | ALA4848002 | 27; CYR715 | Activity | 0 | ALA4815926 | Dose-Dependent Effect | ||||||
| 4. | ALA4848002 | 27; CYR715 | Activity | 0 | ALA4815925 | Not Active | Homo sapiens | |||||
| 5. | ALA4848002 | 27; CYR715 | Activity | 0 | ALA4815924 | Not Active | Homo sapiens | |||||
| 6. | ALA4848002 | 27; CYR715 | Activity | 0 | ALA4815923 | Active | Homo sapiens | |||||
| 7. | ALA4848002 | 27; CYR715 | F | > | 100 | % | ALA4815922 | % | ||||
| 8. | ALA4848002 | 27; CYR715 | AUC | = | 3.7 | hr.microg/ml | ALA4815921 | ng.hr.mL-1 | ||||
| 9. | ALA4848002 | 27; CYR715 | CL | = | 9.2 | ml/min.kg | ALA4815920 | mL.min-1.kg-1 | ||||
| 10. | ALA4848002 | 27; CYR715 | t1/2 | = | 3.5 | hr | ALA4815918 | hr | ||||
| 11. | ALA4848002 | 27; CYR715 | solubility | = | 21 | ug ml-1 | ALA4815916 | ug.mL-1 | ||||
| 12. | ALA4848002 | 27; CYR715 | Papp | = | 40 | 10^-6 cm/s | ALA4815915 | 10^-6 cm/s | ||||
| 13. | ALA4848002 | 27; CYR715 | CLH | = | 63 | microL/min/mg | ALA4815914 | mL.min-1.g-1 | ||||
| 14. | ALA4848002 | 27; CYR715 | Drug metabolism | 0 | ALA4815913 | Metabolite_Detected | ||||||
| 15. | ALA4848002 | 27; CYR715 | CLH | = | 32 | uL/min | ALA4815912 | uL/min | ||||
| 16. | ALA4848002 | 27; CYR715 | EC50 | = | 40 | nM | ALA4815911 | 7.40 | nM | Homo sapiens |
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