# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4848517 | 8 | ED50 | > | 100 | mg kg-1 | ALA5236049 | mg.kg-1 | Mus musculus | |||
2. | ALA4848517 | 8 | IC50 | > | 10 | uM | ALA5236048 | nM | Mus musculus | |||
3. | ALA4848517 | 8 | Emax | = | 57 | % | ALA5236047 | % | Mus musculus | |||
4. | ALA4848517 | 8 | EC50 | = | 3586.3 | nM | ALA5236046 | 5.45 | nM | Mus musculus | ||
5. | ALA4848517 | 8 | Emax | = | 54 | % | ALA5236042 | % | Mus musculus | |||
6. | ALA4848517 | 8 | EC50 | = | 9384 | nM | ALA5236041 | 5.03 | nM | Mus musculus | ||
7. | ALA4848517 | 8 | Ki | = | 3395 | nM | ALA5236040 | 5.47 | nM | Mus musculus | ||
8. | ALA4848517 | 8 | Ki | = | 883.33 | nM | ALA5236039 | 6.05 | nM | Mus musculus | ||
9. | ALA4848517 | 8 | Ki | = | 665.7 | nM | ALA5236038 | 6.18 | nM | Mus musculus | ||
10. | ALA4848517 | 8 | IC50 | = | 10000 | nM | ALA5127645 | 5.00 | nM | Homo sapiens | ||
11. | ALA4848517 | 8 | IC50 | > | 10000 | nM | ALA5127644 | nM | Homo sapiens | |||
12. | ALA4848517 | 8 | IC50 | = | 2200 | nM | ALA5127643 | 5.66 | nM | Homo sapiens | ||
13. | ALA4848517 | 8 | Ki | = | 2560 | nM | ALA5127527 | 5.59 | nM | Homo sapiens | ||
14. | ALA4848517 | 8 | Ki | > | 10000 | nM | ALA5127526 | nM | Homo sapiens | |||
15. | ALA4848517 | 8 | Ki | = | 410 | nM | ALA5127525 | 6.39 | nM | Homo sapiens | ||
16. | ALA4848517 | 8 | Ki | = | 410 | nM | ALA4808365 | 6.39 | nM | Homo sapiens | ||
17. | ALA4848517 | 8 | Drug recovery | > | 80 | % | ALA4834835 | % | ||||
18. | ALA4848517 | 8 | Drug recovery | > | 90 | % | ALA4834834 | % | ||||
19. | ALA4848517 | 8 | Cp | < | 1 | ng/ml | ALA4834829 | ng/ml | ||||
20. | ALA4848517 | 8 | Cp | < | 1 | ng/ml | ALA4834828 | ng/ml |