| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4850904 | 12a; SLU-2633 | Emax | = | 79 | % | ALA4810713 | % | Homo sapiens | |||
| 2. | ALA4850904 | 12a; SLU-2633 | EC50 | = | 7.7 | uM | ALA4810712 | 5.11 | nM | Homo sapiens | ||
| 3. | ALA4850904 | 12a; SLU-2633 | Activity | 0 | ALA4810711 | Active | Cryptosporidium parvum | |||||
| 4. | ALA4850904 | 12a; SLU-2633 | Activity | > | 99 | % | ALA4810710 | % | Cryptosporidium parvum | |||
| 5. | ALA4850904 | 12a; SLU-2633 | F | = | 1 | % | ALA4810709 | % | ||||
| 6. | ALA4850904 | 12a; SLU-2633 | Vd | = | 130 | ml/kg | ALA4810708 | L.kg-1 | ||||
| 7. | ALA4850904 | 12a; SLU-2633 | Vd | = | 62 | ml/kg | ALA4810707 | L.kg-1 | ||||
| 8. | ALA4850904 | 12a; SLU-2633 | CL | = | 42 | ml/hr/kg | ALA4810706 | mL.min-1.kg-1 | ||||
| 9. | ALA4850904 | 12a; SLU-2633 | CL | = | 19 | ml/hr/kg | ALA4810705 | mL.min-1.kg-1 | ||||
| 10. | ALA4850904 | 12a; SLU-2633 | t1/2 | = | 5.4 | hr | ALA4810704 | hr | ||||
| 11. | ALA4850904 | 12a; SLU-2633 | t1/2 | = | 2.2 | hr | ALA4810703 | hr | ||||
| 12. | ALA4850904 | 12a; SLU-2633 | Cmax | = | 36000 | ng/ml | ALA4810702 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 13. | ALA4850904 | 12a; SLU-2633 | Cmax | = | 1500 | ng/ml | ALA4810701 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 14. | ALA4850904 | 12a; SLU-2633 | Cmax | = | 15000 | ng/ml | ALA4810700 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 15. | ALA4850904 | 12a; SLU-2633 | Cmax | = | 17000 | ng/ml | ALA4810699 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 16. | ALA4850904 | 12a; SLU-2633 | AUC | = | 240000 | hr.ng/ml | ALA4810698 | ng.hr.mL-1 | ||||
| 17. | ALA4850904 | 12a; SLU-2633 | AUC | = | 5200 | hr.ng/ml | ALA4810697 | ng.hr.mL-1 | ||||
| 18. | ALA4850904 | 12a; SLU-2633 | AUC | = | 55000 | hr.ng/ml | ALA4810696 | ng.hr.mL-1 | ||||
| 19. | ALA4850904 | 12a; SLU-2633 | AUC | = | 50000 | hr.ng/ml | ALA4810695 | ng.hr.mL-1 | ||||
| 20. | ALA4850904 | 12a; SLU-2633 | Ratio | = | 5.8 | ALA4810694 |
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