# | Name | Compound Key | Action Type | Relation | Activety Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4852096 | 10a | Activity | 0 | ALA4834937 | Not Active | Rattus norvegicus | |||||
2. | ALA4852096 | 10a | Activity | 0 | ALA4834910 | Active | Rattus norvegicus | |||||
3. | ALA4852096 | 10a | Activity | 0 | ALA4834909 | Active | Rattus norvegicus | |||||
4. | ALA4852096 | 10a | Activity | 0 | ALA4834908 | Active | Rattus norvegicus | |||||
5. | ALA4852096 | 10a | AUC | = | 7918 | hr.ng/ml | ALA4834881 | ng.hr.mL-1 | ||||
6. | ALA4852096 | 10a | AUC | = | 3520 | hr.ng/ml | ALA4834879 | ng.hr.mL-1 | ||||
7. | ALA4852096 | 10a | Cmax | = | 6490 | uM | ALA4834878 | nM | ||||
8. | ALA4852096 | 10a | Cmax | = | 3535 | uM | ALA4834876 | nM | ||||
9. | ALA4852096 | 10a | t1/2 | = | 1.42 | hr | ALA4834875 | hr | ||||
10. | ALA4852096 | 10a | t1/2 | = | 0.67 | hr | ALA4834873 | hr | ||||
11. | ALA4852096 | 10a | F | = | 138 | % | ALA4834872 | % | ||||
12. | ALA4852096 | 10a | F | = | 112.3 | % | ALA4834870 | % | ||||
13. | ALA4852096 | 10a | Activity | = | 2052 | ng/ml | ALA4834869 | ng/ml | ||||
14. | ALA4852096 | 10a | Activity | = | 2726 | ng/ml | ALA4834866 | ng/ml | ||||
15. | ALA4852096 | 10a | t1/2 | = | 0.18 | hr | ALA4834865 | hr | ||||
16. | ALA4852096 | 10a | t1/2 | = | 0.14 | hr | ALA4834862 | hr | ||||
17. | ALA4852096 | 10a | Vdss | = | 0.43 | L/Kg | ALA4834861 | L.kg-1 | ||||
18. | ALA4852096 | 10a | Vdss | = | 0.43 | L/Kg | ALA4834858 | L.kg-1 | ||||
19. | ALA4852096 | 10a | CL | = | 29.4 | ml/min.kg | ALA4834856 | mL.min-1.kg-1 | ||||
20. | ALA4852096 | 10a | CL | = | 53.3 | ml/min.kg | ALA4834854 | mL.min-1.kg-1 |