| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA4854446 | 17e | IC50 | = | 4.76 | uM | ALA5224075 | 5.32 | nM | Homo sapiens | ||
| 2. | ALA4854446 | 17e | IC50 | = | 2.13 | uM | ALA5224074 | 5.67 | nM | Homo sapiens | ||
| 3. | ALA4854446 | 17e | IC50 | = | 5.83 | uM | ALA5224073 | 5.23 | nM | Homo sapiens | ||
| 4. | ALA4854446 | 17e | IC50 | = | 3.29 | uM | ALA5224069 | 5.48 | nM | Homo sapiens | ||
| 5. | ALA4854446 | 17e | IC50 | = | 5.5 | uM | ALA5224068 | 5.26 | nM | Homo sapiens | ||
| 6. | ALA4854446 | 17e | IC50 | = | 6 | uM | ALA5224067 | 5.22 | nM | Homo sapiens | ||
| 7. | ALA4854446 | 17e | IC50 | > | 20 | uM | ALA5224066 | nM | ||||
| 8. | ALA4854446 | 17e | IC50 | = | 0.053 | uM | ALA5224065 | 7.28 | nM | Homo sapiens | ||
| 9. | ALA4854446 | 17e | Ratio IC50 | > | 377 | ALA4826374 | ||||||
| 10. | ALA4854446 | 17e | INH | 0 | ALA4826355 | Active | % | Homo sapiens | ||||
| 11. | ALA4854446 | 17e | INH | 0 | ALA4826354 | Active | % | Homo sapiens | ||||
| 12. | ALA4854446 | 17e | INH | 0 | ALA4826353 | Active | % | Homo sapiens | ||||
| 13. | ALA4854446 | 17e | INH | 0 | ALA4826352 | Active | % | Homo sapiens | ||||
| 14. | ALA4854446 | 17e | INH | 0 | ALA4826351 | Active | % | Homo sapiens | ||||
| 15. | ALA4854446 | 17e | Stabilty | = | 56.7 | % | ALA4826350 | % | ||||
| 16. | ALA4854446 | 17e | Stabilty | = | 65.2 | % | ALA4826349 | % | ||||
| 17. | ALA4854446 | 17e | CLH | = | 13.2 | ml/min.kg | ALA4826348 | mL.min-1.kg-1 | ||||
| 18. | ALA4854446 | 17e | CLH | = | 14.6 | microL/min/mg | ALA4826347 | mL.min-1.g-1 | ||||
| 19. | ALA4854446 | 17e | t1/2 | = | 94.7 | min | ALA4826346 | hr | ||||
| 20. | ALA4854446 | 17e | IC50 | = | 4.76 | uM | ALA4826345 | 5.32 | nM | Homo sapiens |
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